Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

被引:2270
|
作者
Meanwell, Nicholas A. [1 ]
机构
[1] Bristol Myers Squibb Pharmaceut Res & Dev, Dept Med Chem, Wallingford, CT 06492 USA
关键词
ADRENOCEPTOR-SELECTIVE ANTAGONISTS; CALCIUM-CHANNEL BLOCKERS; HYDROGEN-BOND BASICITY; CENTER-DOT-O; NONPROSTANOID PROSTACYCLIN MIMETICS; ALPHA-KETOHETEROCYCLIC INHIBITORS; ACTIVE NONPEPTIDIC INHIBITORS; RESPIRATORY SYNCYTIAL VIRUS; ELECTRON-WITHDRAWING POWER; OPIOID AGONIST METABOLITES;
D O I
10.1021/jm1013693
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:2529 / 2591
页数:63
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