共 50 条
- [21] APPROACH TO THE DISCOVERY OF NOVEL, SELECTIVE INHIBITORS OF P56(LCK) TYROSINE KINASE - IDENTIFICATION OF NON-HYDROXYLATED CHROMONES AS P56(LCK) INHIBITORSDRUG DEVELOPMENT RESEARCH, 1995, 34 (04) : 344 - 352MILLER, D论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAWANG, S论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAREID, J论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAXIE, W论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAGAUVIN, B论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAKELLEY, M论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PASARUP, J论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PASAWUTZ, DG论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAMISKI, M论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PADOLLE, RE论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PAFALTYNEK, CR论文数: 0 引用数: 0 h-index: 0机构: STERLING WINTHROP,DEPT IMMUNOL,DIV PHARMACEUT RES,COLLEGEVILLE,PA
- [22] Novel 2-aminopyrimidine carbamates as potent and orally active inhibitors of Lck: Synthesis, SAR, and in vivo antiinflammatory activityJOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (16) : 4981 - 4991Martin, Matthew W.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USANewcomb, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USANunes, Joseph J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAMcGowan, David C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAArmistead, David M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USABoucher, Christina论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USABuchanan, John L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USABuckner, William论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAChai, Lilly论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAElbaum, Daniel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAEpstein, Linda F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAFaust, Theodore论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAFlynn, Shaun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAGallant, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAGore, Anu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAGu, Yan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAHsieh, Faye论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USALee, Josie H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAMetz, Daniela论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAMiddleton, Scot论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAMohn, Deanna论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAMorgenstern, Kurt论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAMorrison, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USANovak, Perry M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAOliveira-dos-Santos, Antonio论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAPowers, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USARose, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USASchneider, Stephen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USASell, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USATudor, Yanyan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USATurci, Susan M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAWelcher, Andrew A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAWhite, Ryan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAZack, Debra论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAZhao, Huilin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAZhu, Li论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAZhu, Xiaotian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAGhiron, Chiara论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAAmouzegh, Patricia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAErmann, Monika论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAJenkins, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAJohnston, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USANapier, Spencer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USAPower, Eoin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02139 USA
- [23] Discovery and development of orally active P38 kinase inhibitors as anti-TNF agentsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U161 - U161Devraj, RV论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Global Res & Dev, Chesterfield, MO 63017 USA Pfizer, Global Res & Dev, Chesterfield, MO 63017 USA
- [24] Discovery of benzoylisoindolines as a novel class of potent, selective and orally active GlyT1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (23) : 6960 - 6965Pinard, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandAlberati, Daniela论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandBender, Markus论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandBorroni, Edilio论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandBrom, Virginie论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandBurner, Serge论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandFischer, Holger论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandHainzl, Dominik论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandHalm, Remy论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandHauser, Nicole论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandJolidon, Synese论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandLengyel, Judith论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandMarty, Hans-Peter论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandMeyer, Thierry论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandMoreau, Jean-Luc论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandMory, Roland论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandNarquizian, Robert论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandNorcross, Roger D.论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandSchmid, Philipp论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandWermuth, Roger论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, SwitzerlandZimmerli, Daniel论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland F Hoffmann La Roche & Co Ltd, Pharmaceut Res Basel, CH-4070 Basel, Switzerland
- [25] Discovery of potent and orally active farnesyltransferase (FT) inhibitors.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U29 - U29Tong, YS论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAWang, L论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAHasvold, L论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALeonard, N论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALi, TM论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALi, Q论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAWang, WB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USACohen, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAGu, WZ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAZhang, HY论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USABauch, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAMarsh, K论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USARosenberg, SH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALin, NH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USASham, HL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA
- [26] The active site of arginine kinase.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1999, 217 : U422 - U422Binz, S论文数: 0 引用数: 0 h-index: 0机构: Loras Coll, Dubuque, IA 52001 USA Loras Coll, Dubuque, IA 52001 USASpeckhard, D论文数: 0 引用数: 0 h-index: 0机构: Loras Coll, Dubuque, IA 52001 USA Loras Coll, Dubuque, IA 52001 USA
- [27] Optimization of 2-phenylaminoimidazo[4,5-h]isoquinolin-9-ones:: Orally active inhibitors of lck kinaseJOURNAL OF MEDICINAL CHEMISTRY, 2003, 46 (08) : 1337 - 1349Goldberg, DR论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAButz, T论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USACardozo, MG论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAEckner, RJ论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAHammach, A论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAHuang, J论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAJakes, S论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAKapadia, S论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAKashem, M论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USALukas, S论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAMorwick, TM论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAPanzenbeck, M论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAPatel, U论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAPav, S论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAPeet, GW论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAPeterson, JD论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAProkopowicz, AS论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USASnow, RJ论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USASellati, R论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USATakahashi, H论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USATan, J论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USATschantz, MA论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAWang, XJ论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAWang, Y论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAWolak, J论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAXiong, P论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USAMoss, N论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharmaceut Inc, Dept Med Chem, Ridgefield, CT 06877 USA
- [28] Synthesis and biological evaluation of a series of novel and potent inhibitors of KDR kinase.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U44 - U44Tucker, TJ论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USACiecko, PA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAColl, KE论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAHartman, GD论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USALumma, WC论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAMerkle, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAMcFall, RC论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAMcGaughey, GB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USARickert, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAShipman, JM论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USASingh, R论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USASisko, JT论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USASmith, AM论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USAThomas, KA论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, W Point, PA 19486 USA
- [29] Discovery of Isonicotinamides as Highly Selective, Brain Penetrable, and Orally Active Glycogen Synthase Kinase-3 InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (03) : 1041 - 1051Luo, Guanglin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAChen, Ling论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USABurton, Catherine R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAXiao, Hong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USASivaprakasam, Prasanna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAKrause, Carol M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USACao, Yang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USALiu, Nengyin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USALippy, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAClarke, Wendy J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USASnow, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USARaybon, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAArora, Vinod论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAPokross, Matt论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAKish, Kevin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USALewis, Hal A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USALangley, David R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAMacor, John E.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USADubowchik, Gene M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Bristol Myers Squibb Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA
- [30] Structure-based drug design:: the discovery of novel nonpeptide orally active inhibitors of human reninCHEMISTRY & BIOLOGY, 2000, 7 (07): : 493 - 504Rahuel, J论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandRasetti, V论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandMaibaum, J论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, Switzerland Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandRüeger, H论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandGöschke, R论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandCohen, NC论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandStutz, S论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandCumin, F论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandFuhrer, W论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandWood, JM论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, SwitzerlandGrütter, MG论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharma AG, Metab & Cardiovasc Dis, CH-4002 Basel, Switzerland