共 50 条
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- [42] Antitumor Efficacy of PKI-587, a Highly Potent Dual PI3K/mTOR Kinase InhibitorCLINICAL CANCER RESEARCH, 2011, 17 (10) : 3193 - 3203Mallon, Robert论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAFeldberg, Larry R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USALucas, Judy论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAChaudhary, Inder论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Drug Safety & Metab, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USADehnhardt, Christoph论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USADelos Santos, Efren论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAChen, Zecheng论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAdos Santos, Osvaldo论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAAyral-Kaloustian, Semiramis论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAVenkatesan, Aranapakam论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Discovery Med Chem, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USAHollander, Irwin论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Dept Oncol, Pearl River, NY 10965 USA Pfizer, Dept Oncol, Pearl River, NY 10965 USA
- [43] The dual PI3K/mTOR inhibitor dactolisib elicits anti-tumor activity in vitro and in vivoONCOTARGET, 2018, 9 (01) : 706 - 717Shi, Fei论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaZhang, Jinying论文数: 0 引用数: 0 h-index: 0机构: Chinese Peoples Liberat Army Gen Hosp, Inst Basic Med Sci, Beijing 100853, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaLiu, Hongyu论文数: 0 引用数: 0 h-index: 0机构: Chinese Peoples Liberat Army Gen Hosp, Key Lab, Canc Ctr, Beijing 100853, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaWu, Liangliang论文数: 0 引用数: 0 h-index: 0机构: Chinese Peoples Liberat Army Gen Hosp, Key Lab, Canc Ctr, Beijing 100853, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaJiang, Hongyu论文数: 0 引用数: 0 h-index: 0机构: Wuxi Third Peoples Hosp, Dept Anesthesiol, Wuxi 214000, Jiangsu, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaWu, Qiyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Peoples Liberat Army Gen Hosp, Key Lab, Canc Ctr, Beijing 100853, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaLiu, Tianyi论文数: 0 引用数: 0 h-index: 0机构: Chinese Peoples Liberat Army Gen Hosp, Key Lab, Canc Ctr, Beijing 100853, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaLou, Meiqing论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R ChinaWu, Hao论文数: 0 引用数: 0 h-index: 0机构: Capital Med Univ, Xuanwu Hosp, Dept Neurosurg, Beijing 100053, Peoples R China Shanghai Jiao Tong Univ, Shanghai Gen Hosp, Dept Neurosurg, Sch Med, Shanghai 200000, Peoples R China
- [44] A dual PI3K/AKT/mTOR signaling inhibitor miR-99a suppresses endometrial carcinomaAMERICAN JOURNAL OF TRANSLATIONAL RESEARCH, 2016, 8 (02): : 719 - 731Li, Yunyun论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R ChinaZhang, Zhongzu论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Yongchuan Hosp, Dept Orthoped, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R ChinaZhang, Xiaojing论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R ChinaLin, Ying论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R ChinaLuo, Tangshu论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R ChinaXiao, Zhenghua论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R ChinaZhou, Qin论文数: 0 引用数: 0 h-index: 0机构: Chongqing Med Univ, Affiliated Hosp 1, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China Chongqing Med Univ, Yongchuan Hosp, Dept Gynecol & Obstet, Chongqing 402160, Peoples R China
- [45] Preclinical efficacy of GNE-317, a dual PI3K/mTOR inhibitor, with or without bevacizumab in EGFR and/or PTEN-mutated glioblastoma multiformeCANCER RESEARCH, 2014, 74 (19)Sio, Terence T.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USAPokorny, Jenny L.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USAMladek, Ann C.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USACarlson, Brett L.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USASchroeder, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USAIyekegbe, Dennis O.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USABakken, Katrina论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Mayo Clin, Rochester, MN USAPhillips, Heidi论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Mayo Clin, Rochester, MN USASarkaria, Jann N.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Mayo Clin, Rochester, MN USA
- [46] Design, synthesis and bioevaluation of novel substituted triazines as potential dual PI3K/mTOR inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 204Wu, Ting-Ting论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaGuo, Qing-Qing论文数: 0 引用数: 0 h-index: 0机构: South China Univ Technol, Guangdong Prov Engn & Technol Res Ctr Biopharmace, Sch Biol & Biol Engn, Joint Int Res Lab Synthet Biol & Med,Minist Educ, Guangzhou 510006, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaChen, Zi-Li论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Affiliated Hosp, Guiyang 550004, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaWang, Li-Li论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaDu, Yao论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaChen, Rui论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaMao, Yuan-Hu论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaYang, Sheng-Gang论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaHuang, Jing论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaWang, Jian-Ta论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaWang, Ling论文数: 0 引用数: 0 h-index: 0机构: South China Univ Technol, Guangdong Prov Engn & Technol Res Ctr Biopharmace, Sch Biol & Biol Engn, Joint Int Res Lab Synthet Biol & Med,Minist Educ, Guangzhou 510006, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaTang, Lei论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R ChinaZhang, Ji-Quan论文数: 0 引用数: 0 h-index: 0机构: Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China Guizhou Med Univ, Coll Pharm, Guizhou Prov Engn Technol Res Ctr Chem Drug R&D, State Key Lab Funct & Applicat Med Plants, Guiyang 550004, Guizhou, Peoples R China
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- [49] The Role of PI3K/mTOR Inhibition in Combination with Sorafenib in Hepatocellular Carcinoma TreatmentANTICANCER RESEARCH, 2012, 32 (07) : 2531 - 2536论文数: 引用数: h-index:机构:Angulo, Paul论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Internal Med, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USAChen, Changguo论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USACreasy, Kate Townsend论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Immunol, Lexington, KY USA Univ Kentucky, Coll Med, Markey Canc Ctr, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USASpear, Brett T.论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Immunol, Lexington, KY USA Univ Kentucky, Coll Med, Markey Canc Ctr, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USAHundley, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USADaily, Michael F.论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USAShah, Malay论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USAEvers, B. Mark论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USA Univ Kentucky, Coll Med, Markey Canc Ctr, Lexington, KY USA Univ Kentucky, Coll Med, Dept Surg, Lexington, KY USA
- [50] Radiosensitization by the Dual PI3K/mTOR inhibitor NVP-BEZ235CANCER RESEARCH, 2012, 72Cerniglia, George J.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAKarar, Jayashree论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAKoumenis, Constantinos论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAMaity, Amit论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USA