Syntheses of Some Thiazolidin-4-ones as Potential Antimicrobial Agents

被引：0
|
作者：
Havaldar, Freddy H. [1 ]
Sharma, Azad Kumar S. [1 ]
机构：
[1] St Xaviers Coll, Nadkarny Sacasa Res Lab, Dept Chem, Bombay 400001, Maharashtra, India
来源：
ASIAN JOURNAL OF CHEMISTRY | 2011年 / 23卷 / 03期
关键词：
Synthesis; Thiazolidin-4-ones; Antibacterial and antifungal activity;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
4-Acetamido-2-methoxybenzoyl hydrazine (1) on condensation with different aromatic aldehydes yielded the substituted benzal-(4'-acetamido-2'-methoxybenzoyl)hydrazines (2a-f) which on cyclization with thioglycolic acid in presence of anhydrous aluminium chloride as catalyst afforded 2-(substituted phenyl)-3-(4'-acetamido-2.-methoxy benzamido)-5-H-thiazolidin-4-ones (3a-f). The structures of the newly synthesized compounds have been established by analytical and spectral methods. These compounds have also been screened for their biological activity.
引用
收藏
页码：1314 / 1316
页数：3
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