Synthesis and evaluation of 18F-labeled 5-(4-piperidinyl)-isothazoles: Imaging the GABA binding site of GABAA receptors

被引:0
|
作者
Vasko, Kramer [1 ]
Vanessa, Bockhardt [2 ]
Helmut, Lueddens [2 ]
Frank, Roesch [1 ]
机构
[1] Johannes Gutenberg Univ Mainz, Inst Nucl Chem, Mainz, Germany
[2] Johannes Gutenberg Univ Mainz, Dept Psychiat, Clin Res Grp, Univ Med Ctr Johannes Gutenberg, D-6500 Mainz, Germany
关键词
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:S285 / S285
页数:1
相关论文
共 50 条
  • [41] Synthesis and in Vitro and in Vivo Evaluation of an 18F-Labeled Neuropeptide Y Analogue for Imaging of Breast Cancer by PET
    Hofmann, Sven
    Maschauer, Simone
    Kuwert, Torsten
    Beck-Sickinger, Annette G.
    Prante, Olaf
    MOLECULAR PHARMACEUTICS, 2015, 12 (04) : 1121 - 1130
  • [42] Synthesis and Evaluation of 18F-Labeled GRP78-Targeting Probe for Prostate Cancer Imaging with PET
    Liu, Shuanglong
    Conti, Peter
    JOURNAL OF NUCLEAR MEDICINE, 2020, 61
  • [43] Synthesis and evaluation of 2-amino-5-(4-[18F]fluorophenyl)pent-4-ynoic acid ([18F]FPhPA): A novel 18F-labeled amino acid for oncologic PET imaging
    Way, Jenilee D.
    Wang, Monica
    Hamann, Ingrit
    Wuest, Melinda
    Wuest, Frank
    NUCLEAR MEDICINE AND BIOLOGY, 2014, 41 (08) : 660 - 669
  • [44] Synthesis and Evaluation of a 18F-Labeled 4-Ipomeanol as an Imaging Agent for CYP4B1 Gene Prodrug Activation Therapy
    Moon, Byung Seok
    Jang, Su Jin
    Kim, Sung Joo
    Lee, Tae Sup
    Chi, Dae Yoon
    Lee, Byung Chul
    Kang, Joo Hyun
    Kim, Sang Eun
    CANCER BIOTHERAPY AND RADIOPHARMACEUTICALS, 2013, 28 (08) : 588 - 597
  • [45] Evaluation of a simple, 18F-labeled radiotracer as PET imaging agent for sigma-1 receptors in the nonhuman primate brain
    Jia, Hongmei
    Cai, Zhengxin
    Holden, Daniel
    He Yingfang
    Lin, Shu-fei
    Li, Songye
    Baum, Evan
    Shirali, Anupama
    Kapinos, Michael
    Gao, Hong
    Ropchan, Jim
    Huang, Yiyun
    JOURNAL OF NUCLEAR MEDICINE, 2018, 59
  • [46] Synthesis and Evaluation of a 18F-Labeled Triazinediamine Analogue for Imaging Mutant IDH1 Expression in Gliomas by PET
    Chitneni, Satish K.
    Yan, Hai
    Zalutsky, Michael R.
    ACS MEDICINAL CHEMISTRY LETTERS, 2018, 9 (07): : 606 - 611
  • [47] Synthesis and evaluation of 4-[18F] fluoropropoxy-3-iodobenzylguanidine ([18F]FPOIBG): A novel 18F-labeled analogue of MIBG
    Vaidyanathan, Ganesan
    McDougald, Darryl
    Koumarianou, Eftychia
    Choi, Jaeyeon
    Hens, Marc
    Zalutsky, Michael R.
    NUCLEAR MEDICINE AND BIOLOGY, 2015, 42 (08) : 673 - 684
  • [48] Synthesis and Biological Evaluation of 18F-labeled FMTPD as a Focal Adhesion Kinase-Targeted Tumor Imaging Agent
    Fang, Yu
    Wang, Dawei
    Xu, Xingyu
    Zhao, Lingzhou
    Zhang, Jinming
    Zhao, Mingxia
    Lu, Xia
    Qi, Chuanmin
    Zhang, Huabei
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2015, 58 : S240 - S240
  • [49] Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents
    Hocke, C
    Prante, O
    Löber, S
    Hübner, H
    Gmeiner, P
    Kuwert, T
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (21) : 4819 - 4823
  • [50] Synthesis and evaluation of 18F-labeled ATP competitive inhibitors of topoisomerase II as probes for imaging topoisomerase II expression
    Daumar, Pierre
    Zeglis, Brian M.
    Ramos, Nicholas
    Divilov, Vadim
    Sevak, Kuntal Kumar
    Pillarsetty, NagaVaraKishore
    Lewis, Jason S.
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 86 : 769 - 781