Non-peptide CRF1 antagonists: Pyrazolo[1,5-a]pyrimidines and pyrazolo[5,1-c][1,2,4]triazines.

被引：0
|
作者：
Wilde, RG
Carter, KL
Klaczkiewicz, JD
Gilligan, PJ
Olson, RE
Zaczek, R
机构：
[1] Dupont Merck Pharmaceut Co, Dept Chem & Phys Sci, Wilmington, DE 19880 USA
[2] Dupont Merck Pharmaceut Co, CNS Dis Res, Wilmington, DE 19880 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2001年 / 221卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
95-MEDI
引用
收藏
页码：U17 / U17
页数：1
相关论文
共 50 条
  • [41] Orally active 3-(3-pyridyl)pyrazolo[1,5-a]pyrimidines as nonpeptide CRF1 receptor antagonists.
    Chen, C
    Wilcoxen, K
    Bozigian, H
    Chen, T
    Cha, M
    McCarthy, JR
    Huang, CQ
    Haddach, M
    Zhu, YF
    Murphy, B
    De Souza, EB
    Grigoriadis, DE
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 221 : U38 - U38
  • [42] Pyrazole-3(5)-diazonium salts in the synthesis of novel pyrazolo[5,1-c][1,2,4]triazines
    Shikhaliev, Kh. S.
    Didenko, V. V.
    Voronkova, V. A.
    Kryl'skii, D. V.
    RUSSIAN CHEMICAL BULLETIN, 2009, 58 (05) : 1034 - 1040
  • [43] Pyrazole-3(5)-diazonium salts in the synthesis of novel pyrazolo[5,1-c][1,2,4]triazines
    Kh. S. Shikhaliev
    V. V. Didenko
    V. A. Voronkova
    D. V. Kryl’skii
    Russian Chemical Bulletin, 2009, 58 : 1034 - 1040
  • [44] Synthesis of some novel pyrazolo[1,5-a]pyrimidine, 1,2,4-triazolo[1,5-a]pyrimidine, pyrido[2,3-d]pyrimidine, pyrazolo[5,1-c]-1,2,4-triazine and 1,2,4-triazolo[5,1-c]-1,2,4-triazine derivatives incorporating a thiazolo[3,2-a]benzimidazole moiety
    Abdel-Aziz, Hatem A.
    Hamdy, Nehal A.
    Farag, Ahmad M.
    Fakhr, Issa M. I.
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2008, 45 (04) : 1033 - 1037
  • [45] Design and Synthesis of Some New Pyrazolo[1,5-a]pyrimidines, Pyrazolo[5,1-c]triazines, Pyrazolo[3,4-d]pyridazines, and Isoxazolo[3,4-d]pyridazines Containing the Pyrazole Moiety
    Abdelhamid, Abdou O.
    Fahmi, Abdelgawad A.
    Halim, Karema N. M.
    SYNTHETIC COMMUNICATIONS, 2013, 43 (08) : 1101 - 1126
  • [46] Chemospecific reactions of as-triazine ring reduction in sulfonyl derivatives of pyrazolo[5,1-c][1,2,4]triazines
    Ledenyova, Irina V.
    Kartavtsev, Pavel A.
    Shikhaliev, Khidmet S.
    Egorova, Alevtina Yu.
    CHEMISTRY OF HETEROCYCLIC COMPOUNDS, 2017, 53 (10) : 1128 - 1133
  • [47] Chemospecific reactions of as-triazine ring reduction in sulfonyl derivatives of pyrazolo[5,1-c][1,2,4]triazines
    Irina V. Ledenyova
    Pavel A. Kartavtsev
    Khidmet S. Shikhaliev
    Alevtina Yu. Egorova
    Chemistry of Heterocyclic Compounds, 2017, 53 : 1128 - 1133
  • [48] RING TRANSFORMATION OF 1,5-BENZOXAZEPINES INTO SPIROBENZOXAZOLES - SYNTHESIS OF PYRAZOLO[1',5'-3,4][1,2,4]TRIAZINO[5,6-B][1,5]BENZOXAZEPINES AND SPIRO[BENZOXAZOLE-2'(3'H),4(1H)PYRAZOLO[5,1-C][1,2,4]TRIAZINES]
    KURASAWA, Y
    OKIYAMA, M
    KAMIGAKI, Y
    KANOH, M
    TAKADA, A
    OKAMOTO, Y
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1988, 25 (04) : 1259 - 1262
  • [49] INTRAMOLECULAR NITRILE IMINE CYCLOADDITIONS TO THE ACETYLENIC BOND IN THE SYNTHESIS OF PYRAZOLO[1,5-A][4,1]-BENZOXAZEPINES AND PYRAZOLO[1,5-A][5,1]BENZOXAZOCINES
    BROGGINI, G
    GARANTI, L
    MOLTENI, G
    ZECCHI, G
    HETEROCYCLES, 1994, 38 (07) : 1601 - 1607
  • [50] Synthesis of Pyrazolo[1,5-a]pyridinyl, Pyrazolo[1,5-a]quinolinyl, and Pyrazolo[5,1-a]isoquinolinyl Sulfonyl Fluorides via a [3+2] Annulation
    Wu, Wen-Qian
    Qin, Hua-Li
    JOURNAL OF ORGANIC CHEMISTRY, 2023, 88 (05): : 3266 - 3276
12345