Reactivity of Substituted 2-Spiropyrimidin-4-Ones Under Vilsmeier-Haack Conditions

被引：5
|
作者：
Varenichenko, S. A. [1 ]
Farat, O. K. [1 ]
Markov, V. I. [1 ]
机构：
[1] Ukrainian State Chem Technol Univ, UA-49005 Dnepropetrovsk, Ukraine
来源：
CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2015年 / 50卷 / 11期
关键词：
hydroacridines; rearrangement; Vilsmeier-Haack reaction; INHIBITORS;
D O I：
10.1007/s10593-014-1626-9
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Substituted 2-spiropyrimidin-4-ones are formylated at room temperature under the conditions of the Vilsmeier-Haack reaction. When cautiously heated they undergo electrophilic rearrangement.
引用
收藏
页码：1602 / 1607
页数：6
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