Synthesis of Imidazo[1,2-c]quinazolin-5(6H)-ones and Benzimidazo[1,2-c]quinazolin-6(5H)-ones with the Aid of Low-Valent Titanium Reagent

被引：14

作者：

Zhao, Xuan ^{[1
]}

Shi, Da-Qing ^{[1
]}

机构：

[1] Soochow Univ, Coll Chem Chem Engn & Mat Sci, Key Lab Organ Synth Jiangsu Prov, Suzhou 215123, Peoples R China

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2010年 / 47卷 / 03期

关键词：

COUPLING REACTIONS; DERIVATIVES; QUINAZOLINES; CYCLIZATIONS;

D O I：

10.1002/jhet.353

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A short and facile synthesis of imidazo[1,2-c]quinazolin-5(6H)-ones and benzimidazo[1,2-c]quinazolin-6(5H)-ones was accomplished in good yields via the novel reductive cyclization of 2-(2-nitrophenyl)-imidazoles or 2-(2-nitrophenyl)benzoimidazoles with isocyanates promoted by low-valent titanium reagent.

引用

页码：524 / 527

页数：4

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