A SMALL-MOLECULE PARP7 INHIBITOR TRIGGERS ANTITUMOR IMMUNITY

被引:1
|
作者
不详
机构
关键词
D O I
10.1158/2159-8290.CD-RW2021-107
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
A small-molecule PARP7 inhibitor caused in vivo tumor regression by restoring interferon signaling. ©2021 American Association for Cancer Research.
引用
收藏
页码:2125 / 2125
页数:1
相关论文
共 50 条
  • [31] The antitumor effect of small molecule inhibitor PSdis
    Cheng, X.
    EUROPEAN JOURNAL OF IMMUNOLOGY, 2019, 49 : 1741 - 1742
  • [32] A new small-molecule Aurora B inhibitor shows antitumor activity in human cancer cell lines
    Yuanyuan Wu
    Jie Li
    Chenxiao Jiang
    Xianmei Yang
    Lihuan Cao
    Long Yu
    Molecular Biology Reports, 2015, 42 : 517 - 524
  • [33] A small-molecule SUMOylation inhibitor activates antitumor immune responses and potentiates immune therapies in preclinical models
    Lightcap, Eric S.
    Yu, Pengfei
    Grossman, Stephen
    Song, Keli
    Khattar, Mithun
    Xega, Kristina
    He, Xingyue
    Gavin, James M.
    Imaichi, Hisashi
    Garnsey, James J.
    Koenig, Erik
    Zhang, Hongru
    Lu, Zhen
    Shah, Pooja
    Fu, Yu
    Milhollen, Michael A.
    Hatton, Beryl A.
    Riceberg, Jessica
    Shinde, Vaishali
    Li, Cong
    Minissale, James
    Yang, Xiaofeng
    England, Dylan
    Klinghoffer, Richard A.
    Langston, Steve
    Galvin, Katherine
    Shapiro, Gary
    Pulukuri, Sai M.
    Fuchs, Serge Y.
    Huszar, Dennis
    SCIENCE TRANSLATIONAL MEDICINE, 2021, 13 (611)
  • [34] Small-molecule PARP modulators - Current status and future therapeutic potential
    Penning, Thomas D.
    CURRENT OPINION IN DRUG DISCOVERY & DEVELOPMENT, 2010, 13 (05) : 577 - 586
  • [35] A new small-molecule Aurora B inhibitor shows antitumor activity in human cancer cell lines
    Wu, Yuanyuan
    Li, Jie
    Jiang, Chenxiao
    Yang, Xianmei
    Cao, Lihuan
    Yu, Long
    MOLECULAR BIOLOGY REPORTS, 2015, 42 (02) : 517 - 524
  • [36] Antitumor Activity and Pharmacodynamic Biomarkers of a Novel and Orally Available Small-Molecule Antagonist of Inhibitor of Apoptosis Proteins
    Sumi, Hiroyuki
    Yabuki, Masato
    Iwai, Kenichi
    Morimoto, Megumi
    Hibino, Ryosuke
    Inazuka, Masakazu
    Hashimoto, Kentaro
    Kosugi, Yohei
    Aoyama, Kazunobu
    Yamamoto, Shunsuke
    Yoshimatsu, Mie
    Yamasaki, Hideki
    Tozawa, Ryuichi
    Ishikawa, Tomoyasu
    Yoshida, Sei
    MOLECULAR CANCER THERAPEUTICS, 2013, 12 (02) : 230 - 240
  • [37] A Whole-Genome CRISPR Screen Identifies AHR Loss as a Mechanism of Resistance to a PARP7 Inhibitor
    Chen, Huadong
    Diolaiti, Morgan E.
    O'Leary, Patrick C.
    Rojc, Ajda
    Krogan, Nevan J.
    Kim, Minkyu
    Ashworth, Alan
    MOLECULAR CANCER THERAPEUTICS, 2022, 21 (07) : 1076 - 1089
  • [38] A Small-Molecule Inhibitor to the Cytokine Interleukin-4
    Quinnell, Sean P.
    Leifer, Becky S.
    Nestor, Stephen T.
    Tan, Kelly
    Sheehy, Daniel F.
    Ceo, Luke
    Doyle, Shelby K.
    Koehler, Angela N.
    Vegas, Arturo J.
    ACS CHEMICAL BIOLOGY, 2020, 15 (10) : 2649 - 2654
  • [39] Supramolecular alleviation of cardiotoxicity of a small-molecule kinase inhibitor
    Yang, Xue
    Huang, Qiaoxian
    Bardelang, David
    Wang, Chunming
    Lee, Simon M. Y.
    Wang, Ruibing
    ORGANIC & BIOMOLECULAR CHEMISTRY, 2017, 15 (38) : 8046 - 8053
  • [40] RAS CAN BE TARGETED BY A MULTIVALENT SMALL-MOLECULE INHIBITOR
    不详
    CANCER DISCOVERY, 2017, 7 (04) : 350 - 350