MEDI 40-Tetrahydro carbazoles: Novel, potent and selective 5-HT6 receptor antagonists

被引：0
|
作者：
Kambhampati, Rama Sastry [1 ]
Konda, Jagadish B. [1 ]
Kothmirkar, Prabhakar [1 ]
Bandyala, Trinath R. [1 ]
Yarra, Sivasekhar N. K. [1 ]
Arepalli, Sobhanadri [1 ]
Shinde, Anil K. [1 ]
Nirogi, Ramakrishna V. S. [1 ]
机构：
[1] Suven Life Sci Ltd, Discovery Res, Hyderabad, Andhra Pradesh 500034, India
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2007年 / 234卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
40-MEDI
引用
下载
收藏
页数：1
相关论文
共 50 条
  • [21] Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists
    Ahmed, M
    Briggs, MA
    Bromidge, SM
    Buck, T
    Campbell, L
    Deeks, NJ
    Garner, A
    Gordon, L
    Hamprecht, DW
    Holland, V
    Johnson, CN
    Medhurst, AD
    Mitchell, DJ
    Moss, SF
    Powles, J
    Seal, JT
    Stean, TO
    Stemp, G
    Thompson, M
    Trail, B
    Upton, N
    Winborn, K
    Witty, DR
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (21) : 4867 - 4871
  • [22] MEDI 41-Novel 1-(arylsulfonyl)-3-(piperidinylmethyl)-1H-indoles as potent and selective 5-HT6 antagonists
    Zhou, Ping
    Li, Yanfang
    Harrison, Boyd L.
    Zhang, Guo Ming
    Smith, Deborah
    Kelly, Michael G.
    Schechter, Lee
    Robichaud, Albert J.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234
  • [23] 1-Sulfonyl-6-Piperazinyl-7-Azaindoles as potent and pseudo-selective 5-HT6 receptor antagonists
    Fabritius, Charles-Henry
    Pesonen, Ullamari
    Messinger, Josef
    Horvath, Raymond
    Salo, Harri
    Galezowski, Michal
    Galek, Mariusz
    Stefanska, Klaudia
    Szeremeta-Spisak, Joanna
    Olszak-Plachta, Marta
    Buda, Anna
    Adamczyk, Justyna
    Krol, Marcin
    Prusis, Peteris
    Sieprawska-Lupa, Magdalena
    Mikulski, Maciej
    Kuokkanen, Katja
    Chapman, Hugh
    Obuchowicz, Radoslaw
    Korjamo, Timo
    Jalava, Niina
    Nowak, Mateusz
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (11) : 2610 - 2615
  • [24] IDENTIFICATION OF NOVEL INDANYLAMIDINOHYDRAZONES AS 5-HT6 ANTAGONISTS
    Mesquida, Neus
    Lopez-Perez, Sara
    Dinares, Immaculada
    Frigola, Jordi
    Merce, Ramon
    Holenz, Joerg
    Perez, Raquel
    Burgueno, Javier
    Alcalde, Ermitas
    DRUGS OF THE FUTURE, 2009, 34 : 126 - 126
  • [25] Tetrahydrocarbazole derivatives as novel and selective 5-HT6 receptor ligands
    Konda, Jagadishbabu
    Kambhampati, Ramasastry
    Kothmirkar, Prabhakar
    Arepalli, Sobhanadri
    Bandyala, Trinath Reddy
    Gudla, Parandhama
    Shinde, Anil K.
    Nirogi, Ramakrishna
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238
  • [26] Amino aryl sulfonamides as novel and potent 5-ht6 receptor ligands
    Nirogi, Ramakrishna
    Kambhampati, Ramasastry
    Bandyala, Trinathreddy
    Konda, Jagadishbabu
    Arepalli, Sobhanadri
    Reballi, Veena
    Kothmirkar, Prabhakar
    Pamuleti, Narasimhareddy G.
    Shinde, Anil
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240
  • [27] Tricyclic azepine derivatives as selective brain penetrant 5-HT6 receptor antagonists
    Trani, Giancarlo
    Baddeley, Stuart M.
    Briggs, Michael A.
    Chuang, Tsu T.
    Deeks, Nigel J.
    Johnson, Christopher N.
    Khazragi, Abir A.
    Mead, Tania L.
    Medhurst, Andrew D.
    Milner, Peter H.
    Quinn, Leann P.
    Ray, Alison M.
    Rivers, Dean A.
    Stean, Tania O.
    Stemp, Geoffrey
    Trail, Brenda K.
    Witty, David R.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (20) : 5698 - 5700
  • [28] Synthesis and pharmacological evaluation of aryl aminosulfonamide derivatives as potent 5-HT6 receptor antagonists
    Nirogi, Ramakrishna V. S.
    Daulatabad, Anand V.
    Parandhama, G.
    Mohammad, Shaikh
    Sastri, K. R.
    Shinde, Anil K.
    Dubey, P. K.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (15) : 4440 - 4443
  • [29] Characterisation of SB-271046, a potent and selective 5-HT6 receptor antagonist
    Routledge, C
    Price, GW
    Bromidge, SM
    Moss, SF
    Newman, H
    Riley, G
    Gager, T
    Brown, AM
    Lightowler, S
    Middlemiss, DN
    BRITISH JOURNAL OF PHARMACOLOGY, 1999, 127 : U16 - U16
  • [30] New aryl sulfonamides compounds as potent and selective 5-ht6 receptor ligands
    Shinde, Anil
    Reballi, Veena
    Tiriveedhi, Vinay
    Gudla, Parandhama
    Kota, Laxman
    Chindhe, Anil
    Rambabu, Namala
    Kambhampati, Ramasastry
    Nirogi, Ramakrishna
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240
12345