Solid phase synthesis of 1,2-disubstituted alkenes: A novel alkynyldihydropyridine to alkenylpyridine isomerization

被引:5
|
作者
Chen, CX [1 ]
Wang, BW [1 ]
Munoz, B [1 ]
机构
[1] Merck Res Labs, San Diego, CA 92131 USA
关键词
solid-phase synthesis; 1,2-disubstituted alkenes; alkynyldihydropyridine; alkenylpyridine; isomerization;
D O I
10.1055/s-2003-43343
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A series of 1,2-disubstituted pyridylalkenes have been prepared using a solid-phase resin approach. This approach takes advantage of a novel alkynyldihydropyridine to alkenylpyridine isomerization.
引用
收藏
页码:2404 / 2406
页数:3
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