Synthesis and antimicrobial activity of 3,4-bis(arylthio)maleimides

被引：10

作者：

Panov, Alexey A. ^{[1
]}

Lavrenov, Sergey N. ^{[1
]}

Simonov, Alexander Y. ^{[1
]}

Mirchink, Elena P. ^{[1
]}

Isakova, Elena B. ^{[1
]}

Trenin, Alexey S. ^{[1
]}

机构：

[1] Gause Inst New Antibiot, 11 B Pirogovskaya St, Moscow 119021, Russia

来源：

JOURNAL OF ANTIBIOTICS | 2019年 / 72卷 / 02期

基金：

俄罗斯科学基金会;

关键词：

TEICOPLANIN PSEUDOAGLYCON DERIVATIVES; MALEIMIDES; INHIBITORS;

D O I：

10.1038/s41429-018-0122-3

中图分类号：

Q81 [生物工程学（生物技术）]; Q93 [微生物学];

学科分类号：

071005 ; 0836 ; 090102 ; 100705 ;

摘要：

A series of 3,4-bis(arylthio)maleimides were synthesized and their antimicrobial activity was evaluated against Gram-positive and Gram-negative bacteria, including multidrug resistant (MDR) strains and some fungi. Most compounds turned out to be highly active, activity being dependent on substituents on phenyl rings.

引用

页码：122 / 124

页数：3

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