Development of historic deacetylase inhibitors.

被引:0
|
作者
Richon, VM [1 ]
机构
[1] Aton Pharma Inc, Tarrytown, NY USA
关键词
D O I
暂无
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:6272S / 6272S
页数:1
相关论文
共 50 条
  • [41] Benzofused hydroxamic acids: Useful fragments for the preparation of histone deacetylase inhibitors. Part 1: Hit identification
    Marastoni, Elena
    Bartoli, Sandra
    Berettoni, Marco
    Cipollone, Amalia
    Ettorre, Alessandro
    Fincham, Christopher I.
    Mauro, Sandro
    Paris, Marielle
    Porcelloni, Marina
    Bigioni, Mario
    Binaschi, Monica
    Nardelli, Federica
    Parlani, Massimo
    Maggi, Carlo A.
    Fattori, Daniela
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (14) : 4091 - 4095
  • [42] Development of neutral phosphotyrosine mimetics as protein tyrosine phosphatase inhibitors.
    Wess, J
    Li, B
    Hamdan, FF
    Brichta, L
    Nowak, N
    Bloodworth, L
    Schmidt, C
    Han, SJ
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2004, 227 : U43 - U43
  • [43] Anti-tumoral efficacy of four different historic deacetylase inhibitors on hepatoma cells in vitro
    Ganslmayer, M
    Herold, C
    Ocker, M
    Hahn, E
    Schuppan, D
    GASTROENTEROLOGY, 2003, 124 (04) : A567 - A567
  • [44] Development of an in vivo model to test chondroprotection by selective MMP inhibitors.
    Goldberg, RL
    Doughty, J
    Haston, W
    Blancuzzi, V
    Singh, HN
    Ganu, V
    Melton, R
    Koehn, J
    Skiles, J
    Monovich, L
    Fink, C
    McQuire, L
    O'Byrne, E
    ARTHRITIS AND RHEUMATISM, 1999, 42 (09): : S253 - S253
  • [45] Development and characterization of small molecule HPK1 inhibitors.
    Kujawa, Maciej
    Zimolag, Eliza
    Galezowski, Michal
    Guzik, Pawel
    Dudek, Agata
    Gondela, Andrzej
    Nowogrodzki, Marcin
    Girardi, Marianna
    Krolenko, Kostiantyn
    Bugaj, Marta
    Sudol, Sylwia
    Gibas, Agnieszka
    Szeremeta-Spisak, Joanna
    Bobowska, Aneta
    Zastawna, Magdalena
    Wyrebek, Przemyslaw
    Boutard, Nicolas
    Wieckowska, Aleksandra
    Jasnosz, Wojciech
    Schonemann, Wojciech
    Zuchowicz, Karol
    Synak, David
    Kulesza, Urszula
    Leventes, Oleksandr
    Swirski, Mateusz
    Sasmal, Sujit
    Gluza, Karolina
    Kret, Patryk
    Ogorek, Mateusz
    Michalik, Kinga
    Banaszak, Katarzyna
    Podkowa, Adrian
    Wnuk-Lipinska, Katarzyna
    Dobrzanska, Monika
    Littlewood, Peter
    Brzozka, Krzysztof
    Bartosik, Anna
    Chmielewski, Stefan
    CANCER RESEARCH, 2021, 81 (13)
  • [46] Development of potent, selective and orally available factor Xa inhibitors.
    Shaw, KJ
    Arnaiz, DO
    Buckman, BO
    Chou, YL
    Davey, DD
    Eagen, K
    Griedel, BD
    Guilford, WJ
    Kochanny, M
    Mohan, R
    Ng, H
    Phillips, GB
    Pinkerton, M
    Sakata, S
    Wu, SC
    Xu, W
    Yun, W
    Zhao, Z
    Light, D
    Dallas, J
    Koovakkat, S
    Whitlow, M
    Liang, A
    Trinh, L
    Ho, E
    Smith, D
    Subramanyam, B
    Vergona, R
    Walters, J
    White, KA
    Sullivan, ME
    Morrissey, MM
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1998, 215 : U919 - U919
  • [47] DNA topoisomerases and their inhibitors.
    Pommier, Y
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 211 : 25 - CARB
  • [48] Corrosion inhibitors. A review
    Kadhim, A.
    Al-Amiery, A. A.
    Alazawi, R.
    Al-Ghezi, M. K. S.
    Abass, R. H.
    INTERNATIONAL JOURNAL OF CORROSION AND SCALE INHIBITION, 2021, 10 (01): : 54 - 67
  • [49] Tyrosine kinase inhibitors.
    He, W
    Myers, MR
    Spada, AP
    Hanney, BA
    Setzer, N
    Mailliet, P
    Gontier, S
    Guegen, JC
    Cans, P
    Orton, E
    Cheve, M
    Kubiak, GG
    Shah, HG
    O'Brien, MK
    Bilder, GE
    Allen, E
    Bissery, MC
    Page, K
    Natarajan, C
    Jayyosi, Z
    Kelley, MF
    Toutain, H
    Constan, A
    Amin, D
    Needle, S
    Galczenski, H
    Wang, W
    Perrone, MH
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 219 : U57 - U57
  • [50] SULPHONATES AS RUST INHIBITORS.
    Anand, O.N.
    Malik, V.P.
    Neemla, K.D.
    Kumar, Vijayu
    Anti-Corrosion Methods and Materials, 1986, 33 (07) : 12 - 18