ω-iodoalkyl(methyl)malonate esters

被引：0
|
作者：
Bendler, SE [1 ]
Bundy, JS [1 ]
Clark, SA [1 ]
Davis, DN [1 ]
Orwar, NA [1 ]
Chesnut, RW [1 ]
机构：
[1] Eastern Illinois Univ, Dept Chem, Charleston, IL 61920 USA
来源：
SYNTHETIC COMMUNICATIONS | 2003年 / 33卷 / 19期
关键词：
malonate esters; bioconjugate;
D O I：
10.1081/SCC-120023994
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
omega-Iodoalkyl(methyl)malonate esters have potential utility in the bio-conjugate chemistry of steroids. A representative set of these esters with a variety of protecting groups and alkyl groups has been prepared. The compounds offer a range of elution values on silica, as well as several convenient deprotection options.
引用
收藏
页码：3365 / 3371
页数：7
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