Direct synthesis of Fmoc protected amino acid hydroxamates from acid chlorides mediated by magnesium oxide

被引：14
|
作者：
Vasanthakumar, GR [1 ]
Babu, VVS [1 ]
机构：
[1] Bangalore Univ, Dept Studies Chem, Bangalore 560001, Karnataka, India
来源：
TETRAHEDRON LETTERS | 2003年 / 44卷 / 21期
关键词：
D O I：
10.1016/S0040-4039(03)00830-X
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The synthesis of Fmoc protected amino acid hydroxamates using Fmoc-amino acid chlorides and magnesium oxide is described. The method is simple and efficient, results in complete conversion, and gives good yields and satisfactory purity. (C) 2003 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：4099 / 4101
页数：3
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