Novel nonsteroidal progesterone receptor antagonists derived from thalidomide

被引：0
|
作者：
Nakagawa, Aya
Tanatani, Aya
Miyachi, Hiroyuki
Hashimoto, Yuichi
机构：
[1] Univ Tokyo, Inst Mol & Cellular Biosci, Bunkyo Ku, Tokyo 1130032, Japan
[2] Ochanomizu Univ, Fac Sci, Bunkyo Ku, Tokyo 1128610, Japan
来源：
DRUGS OF THE FUTURE | 2007年 / 32卷
关键词：
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：92 / 93
页数：2
相关论文
共 50 条
  • [31] Nonsteroidal progesterone receptor ligands with unprecedented receptor selectivity
    Palmer, S
    Campen, CA
    Allan, GF
    Rybczynski, P
    Haynes-Johnson, D
    Hutchins, A
    Kraft, P
    Kiddoe, M
    Lai, MT
    Lombardi, E
    Pedersen, P
    Hodgen, G
    Combs, DW
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 2000, 75 (01): : 33 - 42
  • [32] COMP 58-Identification of a potent novel nonsteroidal progesterone receptor modulator from a virtual screen
    Unwalla, Ray J.
    Fensome, Andrew
    Marella, Michael
    Cross, Jason
    Melenski, Edward
    Wilhelm, James
    Olland, Andrea
    Wolfrom, Scott
    Elokdah, Hassan
    Wrobel, Jay
    Winneker, Richard C.
    Yudt, Matthew
    Nagpal, Sunil
    Cohen, Jeff
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2008, 235
  • [33] Discovery and preliminary SAR studies of a novel, nonsteroidal progesterone receptor antagonist pharmacophore
    Pooley, CLF
    Edwards, JP
    Goldman, ME
    Wang, MW
    Marschke, KB
    Crombie, DL
    Jones, TK
    JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (18) : 3461 - 3466
  • [34] Structural development of liver X receptor (LXR) antagonists derived from thalidomide-related glucosidase inhibitors
    Noguchi-Yachide, Tornorru
    Miyachi, Hiroyuki
    Aoyama, Hiroshi
    Aoyama, Atsushl
    Makishima, Makoto
    Hashimoto, Yuichi
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2007, 55 (12) : 1750 - 1754
  • [35] Synthesis and pharmacological evaluation of novel arylpiperazine derivatives as nonsteroidal androgen receptor antagonists
    Kinoyama, I
    Taniguchi, N
    Yoden, T
    Koutoku, H
    Furutani, T
    Kudoh, M
    Okada, M
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2004, 52 (11) : 1330 - 1333
  • [36] Design and synthesis of nonsteroidal progesterone receptor antagonists based on C,C′-diphenylcarborane scaffold as a hydrophobic pharmacophore
    Fujii, Shinya
    Yamada, Ayumi
    Nakano, Eiichi
    Takeuchi, Yuki
    Mori, Shuichi
    Masuno, Hiroyuki
    Kagechika, Hiroyuki
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 84 : 264 - 277
  • [37] Triterpenes from Alisma orientalis act as androgen receptor agonists, progesterone receptor antagonists, and glucocorticoid receptor antagonists
    Lin, Hsiang-Ru
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (15) : 3626 - 3632
  • [38] Novel antagonists of the inhibitory glycine receptor derived from quinolinic acid compounds
    Schmieden, V
    Jezequel, S
    Betz, H
    MOLECULAR PHARMACOLOGY, 1996, 50 (05) : 1200 - 1206
  • [39] Synthesis and identification of novel oxa-steroids as progesterone receptor antagonists
    Kang, Fu-An
    Allan, George
    Guan, Jihua
    Jain, Nareshkumar
    Linton, Olivia
    Tannenbaum, Pamela
    Xu, Jun
    Zhu, Peifang
    Gunnet, Joseph
    Chen, Xin
    Demarest, Keith
    Lundeen, Scott
    Sui, Zhihua
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (04) : 907 - 910
  • [40] NOVEL CLASS OF NON-NMDA RECEPTOR ANTAGONISTS DERIVED FROM AMPA
    BREHM, L
    EBERT, B
    MADSEN, U
    CHRISTENSEN, IT
    KROGSGAARDLARSEN, P
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1991, 201 : 30 - MEDI
12345