Synthesis and applications of a novel polymer-supported EEDQ reagent

被引：7
|
作者：
Kakarla, Ramesh [1 ]
Li, Guo [1 ]
Gerritz, Samuel W. [1 ]
机构：
[1] Bristol Myers Squibb Co, Wallingford, CT 06492 USA
来源：
JOURNAL OF COMBINATORIAL CHEMISTRY | 2007年 / 9卷 / 05期
关键词：
D O I：
10.1021/cc070020y
中图分类号：
O69 [应用化学];
学科分类号：
081704 ;
摘要：
A simple synthetic protocol for a novel polymer-supported EEDQ reagent is reported. This reagent promotes solution-phase amide bond formation without any additives or base, as well as the selective coupling of aliphatic amines with acids in the presence of aromatic amines.
引用
收藏
页码：745 / 747
页数：3
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