Phosphonate-containing analogs of cholesteryl ester as novel inhibitors of cholesteryl ester transfer protein

被引：5
|
作者：
Pietzonka, T
Damon, R
Russell, M
Wattanasin, S
机构：
[1] SANDOZ PHARMACEUT CORP,SANDOZ RES INST,PRECLIN RES,DEPT ONCOL,E HANOVER,NJ 07936
[2] SANDOZ PHARMACEUT CORP,SANDOZ RES INST,PRECLIN RES,DEPT METAB DIS,E HANOVER,NJ 07936
[3] SANDOZ PHARMA AG,PRECLIN RES,CH-4002 BASEL,SWITZERLAND
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 16期
关键词：
D O I：
10.1016/0960-894X(96)00350-2
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A series of phosphorus-containing analogs of cholesteryl ester have been synthesized as potential inhibitors of cholesteryl ester transfer protein (CETP). The most potent inhibitor, phosphonate 7, represents a novel inhibitor of CETP. Copyright (C) 1996 Elsevier Science Ltd
引用
收藏
页码：1951 / 1954
页数：4
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