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- [21] Optimization of a novel kinase inhibitor scaffold for the dual inhibition of JAK2 and FAK kinasesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (01) : 133 - 137Zificsak, Craig A.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAGingrich, Diane E.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USABreslin, Henry J.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USADunn, Derek D.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAMilkiewicz, Karen L.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USATheroff, Jay P.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAThieu, Tho V.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAUnderiner, Ted L.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAWeinberg, Linda R.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAimone, Lisa D.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAlbom, Mark S.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAMason, Jennifer L.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USASaville, Lisa论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAHusten, Jean论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAngeles, Thelma S.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAFinn, James P.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAJan, Mahfuza论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAO'Kane, Teresa M.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USADobrzanski, Pawel论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USADorsey, Bruce D.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA
- [22] AT9283, a potent inhibitor of the Aurora kinases and Jak2, has therapeutic potential in myeloproliferative disordersBRITISH JOURNAL OF HAEMATOLOGY, 2010, 150 (01) : 46 - 57Dawson, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Cambridge Inst Med Res, Dept Haematol, Cambridge CB2 1TN, England Univ Cambridge, NHS Trust, Addenbrookes Hosp, Cambridge CB2 1TN, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandCurry, Jayne E.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, England论文数: 引用数: h-index:机构:Beer, Philip A.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Cambridge Inst Med Res, Dept Haematol, Cambridge CB2 1TN, England Univ Cambridge, NHS Trust, Addenbrookes Hosp, Cambridge CB2 1TN, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandGraham, Brent论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandLyons, John F.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandRichardson, Caroline J.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandScott, Mike A.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, NHS Trust, Addenbrookes Hosp, Cambridge CB2 1TN, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandSmyth, Tomoko论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandSquires, Matthew S.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandThompson, Neil T.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandGreen, Anthony R.论文数: 0 引用数: 0 h-index: 0机构: Univ Cambridge, Cambridge Inst Med Res, Dept Haematol, Cambridge CB2 1TN, England Univ Cambridge, NHS Trust, Addenbrookes Hosp, Cambridge CB2 1TN, England Astex Therapeut Ltd, Cambridge CB4 0QA, EnglandWallis, Nicola G.论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut Ltd, Cambridge CB4 0QA, England Astex Therapeut Ltd, Cambridge CB4 0QA, England
- [23] Effects of CYT387, a Potent Novel JAK2 Inhibitor on JAK2-V617F Induced MPDBLOOD, 2008, 112 (11) : 316 - 317Bumm, Thomas G. P.论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USATyner, Jeffrey W.论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Inst Canc, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USADeininger, Jutta论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Inst Canc, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USALoriaux, Marc论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Inst Canc, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USAVanDyke, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Inst Canc, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USADruker, Brian J.论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Inst Canc, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USABurns, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Cytopia Res Pty Ltd, Melbourne, Vic, Australia Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USAFantino, Emmanuelle论文数: 0 引用数: 0 h-index: 0机构: Cytopia Res Pty Ltd, Melbourne, Vic, Australia Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USADeininger, Michael W. N.论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Inst Canc, Portland, OR 97201 USA Oregon Hlth & Sci Univ, Ctr Hematol Malignancies, Portland, OR 97201 USA
- [24] Z3, a novel Jak2 tyrosine kinase small-molecule inhibitor that suppresses Jak2-mediated pathologic cell growthMOLECULAR CANCER THERAPEUTICS, 2008, 7 (08) : 2308 - 2318Sayyah, Jacqueline论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USAMagis, Andrew论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USAOstrov, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Pathol, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Immunol, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Lab Med, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USAAllan, Robert W.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Pathol, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Immunol, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Lab Med, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USABraylan, Raul C.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Pathol, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Immunol, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Lab Med, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USASayeski, Peter P.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA
- [25] Identification of a novel inhibitor of JAK2 tyrosine kinase by structure-based virtual screeningBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (13) : 3598 - 3601Robert Kiss论文数: 0 引用数: 0 h-index: 0机构: Semmelweis Univ, Dept Pharmaceut Chem, H-1092 Budapest, Hungary Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryTimea Polgar论文数: 0 引用数: 0 h-index: 0机构: Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryKirabo, Annet论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungarySayyah, Jacqueline论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryFigueroa, Nicholas C.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryList, Alan F.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Malignant Hematol Program, Tampa, FL 33612 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungarySokol, Lubomir论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Malignant Hematol Program, Tampa, FL 33612 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryZuckerman, Kenneth S.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Malignant Hematol Program, Tampa, FL 33612 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryGali, Meghanath论文数: 0 引用数: 0 h-index: 0机构: Univ S Florida, Dept Chem, Tampa, FL 33620 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryBisht, Kirpal S.论文数: 0 引用数: 0 h-index: 0机构: Univ S Florida, Dept Chem, Tampa, FL 33620 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungarySayeski, Peter P.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, HungaryKeseru, Gyorgy M.论文数: 0 引用数: 0 h-index: 0机构: Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, Hungary Budapest Univ Technol & Econ, Dept Gen & Analyt Chem, H-1111 Budapest, Hungary
- [26] A selective and potent oral inhibitor of the JAK2 tyrosine kinase reverses polycythemia and leukocytosis induced by JAK2V617F in a mouse modelBLOOD, 2007, 110 (11) : 171A - 171AZaleskas, Virginia M.论文数: 0 引用数: 0 h-index: 0机构: Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USAChan, Wayne W.论文数: 0 引用数: 0 h-index: 0机构: Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USAEvangelista, Peter论文数: 0 引用数: 0 h-index: 0机构: Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USALazarides, Katherine论文数: 0 引用数: 0 h-index: 0机构: Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USAChopra, Rajesh论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Res & Dev Boston, Waltham, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USAZinda, Michael论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Res & Dev Boston, Waltham, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USAHuszar, Dennis论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Res & Dev Boston, Waltham, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USAVan Etten, Richard A.论文数: 0 引用数: 0 h-index: 0机构: Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USA Tufts Univ New England Med Ctr, Mol Oncol Res Inst, Boston, MA USA
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- [30] JAK2 inhibitor blocks the inflammation and development of esophageal squamous carcinoma in vitro through JAK/STAT3 signaling pathwayEUROPEAN JOURNAL OF CANCER, 2013, 49 : S581 - S581Fang, J.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaChu, L.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaLi, C.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaHu, F.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaZhang, X.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaChen, Y.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaZhao, H.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R ChinaXu, Q.论文数: 0 引用数: 0 h-index: 0机构: Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China Shanghai Tenth Peoples Hosp, Shanghai, Peoples R China