PHARMACOLOGICAL CHARACTERIZATION OF A HISTONE DEACETYLASE INHIBITOR AND TUMOR CELL-GROWTH INHIBITION PROPERTIES OF NEW BENZOFURANONE COMPOUNDS

被引:0
|
作者
Blanquart, Christophe [1 ]
Francois, Manon [1 ]
Charrier, Cedric [2 ]
Bertrand, Philippe [2 ]
Gregoire, Marc [1 ]
机构
[1] INSERM, U892, F-75654 Paris 13, France
[2] CNRS, Umr 6514, F-75700 Paris, France
关键词
Cancer; HDAC inhibitors; BRET;
D O I
暂无
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:S924 / S924
页数:1
相关论文
共 50 条
  • [21] Entinostat: A novel class I isoform selective histone deacetylase inhibitor (HDACi) with unique pharmacological properties
    Ordentlich, Peter
    Lee, Gloria
    Kunkel, Lori
    Sausville, Edward
    MOLECULAR CANCER THERAPEUTICS, 2009, 8 (12)
  • [22] ACY 1215, A HISTONE DEACETYLASE 6 INHIBITOR, INHIBITS CANCER CELL GROWTH IN MELANOMA
    Wang, F.
    Zhong, B.
    Zhao, Z.
    JOURNAL OF BIOLOGICAL REGULATORS AND HOMEOSTATIC AGENTS, 2018, 32 (04): : 851 - 858
  • [23] Inhibition of human B-cell development into plasmablasts by histone deacetylase inhibitor valproic acid
    Kienzler, Anne-Kathrin
    Rizzi, Marta
    Reith, Maike
    Nutt, Stephen L.
    Eibel, Hermann
    JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 2013, 131 (06) : 1695 - 1699
  • [24] HUMAN-TUMOR CELL-GROWTH INHIBITION BY A HUMAN TUMOR-DERIVED GLYCOPROTEIN
    FUNKHOUSER, WK
    NECKERS, LM
    AMES, RS
    ROTH, JA
    SURGICAL FORUM, 1984, 35 : 394 - 396
  • [25] Cell growth inhibition by the Mad/Max complex through recruitment of histone deacetylase activity
    Sommer, A
    Hilfenhaus, S
    Menkel, A
    Kremmer, E
    Seiser, C
    Loidl, P
    Luscher, B
    CURRENT BIOLOGY, 1997, 7 (06) : 357 - 365
  • [26] Proteomic analysis of pancreatic endocrine tumor cell lines treated with the histone deacetylase inhibitor trichostatin A
    Cecconi, Daniela
    Donadelli, Massimo
    Rinalducci, Sara
    Zolla, Lello
    Scupoli, Maria Teresa
    Scarpa, Aldo
    Palmieri, Marta
    Righetti, Pier Giorgio
    PROTEOMICS, 2007, 7 (10) : 1644 - 1653
  • [27] INHIBITION OF CELL-GROWTH BY COMBINATION OF ALPHA-DIFLUOROMETHYLORNITHINE AND AN INHIBITOR OF SPERMINE SYNTHASE
    HE, Y
    SHIMOGORI, T
    KASHIWAGI, K
    SHIRAHATA, A
    IGARASHI, K
    JOURNAL OF BIOCHEMISTRY, 1995, 117 (04): : 824 - 829
  • [28] INHIBITION OF BREAST-CANCER CELL-GROWTH INVITRO BY A TYROSINE KINASE INHIBITOR
    REDDY, KB
    MANGOLD, GL
    TANDON, AK
    YONEDA, T
    MUNDY, GR
    ZILBERSTEIN, A
    OSBORNE, CK
    CANCER RESEARCH, 1992, 52 (13) : 3636 - 3641
  • [29] Celastrol acts as a new histone deacetylase inhibitor to inhibit colorectal cancer cell growth via regulating macrophage polarity
    Wang, Shuren
    Hu, Guanghui
    Chen, Lechuang
    Ma, Kai
    Hu, Chenfei
    Zhu, Hongxia
    Xu, Ningzhi
    Zhou, Changchun
    Liu, Mei
    CELL BIOLOGY INTERNATIONAL, 2023, 47 (02) : 492 - 501
  • [30] INHIBITION OF CELL SURVIVAL, TUMOR GROWTH AND HISTONE DEACETYLASE (HDAC) ACTIVITY BY THE DIETARY FLAVONOID LUTEOLIN IN HUMAN EPITHELIOID CANCER CELLS
    Iratni, R.
    Attoub, S.
    Hassan, A. H.
    Vanhoecke, B.
    Gaben, A. M.
    Bracke, M.
    Al-Sultan, M.
    Arafat, K.
    Gespach, C.
    Petroianu, G.
    JOURNAL OF THORACIC ONCOLOGY, 2010, 5 (05) : S114 - S114