In vivo and in vitro characterization of azd9343, a novel GABAB receptor agonist and reflux inhibitor

被引：0
|
作者：
Lehmann, Anders
Elebring, Thomas
Jensen, Jorgen
Mattsson, Jan P.
Nilsson, Karolina A.
Saransaari, Pigo
von Unge, Sverker
机构：
来源：
GASTROENTEROLOGY | 2008年 / 134卷 / 04期
关键词：
D O I：
暂无
中图分类号：
R57 [消化系及腹部疾病];
学科分类号：
摘要：
引用
收藏
页码：A131 / A132
页数：2
相关论文
共 50 条
  • [41] AZD5153, a novel BRD4 inhibitor, suppresses human thyroid carcinoma cell growth in vitro and in vivo
    Xu, Kun
    Chen, Dexuan
    Qian, Dong
    Zhang, Shihu
    Zhang, Yi
    Guo, Song
    Ma, Zhaoqun
    Wang, Shui
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2018, 499 (03) : 531 - 537
  • [42] Discovery and in vitro and in vivo characterization of a novel, small-molecule Ras inhibitor class
    Keeton, Adam B.
    Zhu, Bing
    Lee, Kevin J.
    Canzoneri, Joshua C.
    Sigler, Sara C.
    Lindsey, Ashley S.
    Ramirez-Alcantara, Veronica
    Barnes, Luciana
    Mattox, Tyler E.
    McConnell, Kate
    Berry, Kristy L.
    Valiyaveettil, Jacob
    Chen, Xi
    Boyd, Michael R.
    Piazza, Gary A.
    CANCER RESEARCH, 2016, 76
  • [43] In vitro and in vivo characterization of PA01, a novel promising triple reuptake inhibitor
    Hou, Jian
    Xing, Yanli
    Zuo, Daiying
    Wu, Yingliang
    Tian, Jingwei
    Meng, Qingguo
    Yang, Mina
    PHYSIOLOGY & BEHAVIOR, 2015, 138 : 141 - 149
  • [44] In vitro and in vivo characterization of the agonist-dependent D3 dopamine receptor tolerance property
    Cote, Samantha R.
    Kuzhikandathil, Eldo V.
    NEUROPHARMACOLOGY, 2014, 79 : 359 - 367
  • [45] In vitro and in vivo characterization of the selective toll-like receptor 8 agonist GS-9688
    Daffis, S.
    Ramakrishnan, D.
    Niu, C.
    Zheng, J.
    Santos, R.
    Mish, M.
    Chin, G.
    Aktoudianakis, V.
    Metobo, S.
    Pyun, H-J
    Yu, H.
    Lee, G.
    Palazzo, A.
    Frey, C.
    Pflanz, S.
    Delaney, W. E.
    Fletcher, S. P.
    Mackman, R.
    JOURNAL OF HEPATOLOGY, 2017, 66 (01) : S694 - S694
  • [46] Novel Agonist of Adenosine Receptor Induces Relaxation of Corpus Cavernosum in Guinea Pigs: An In Vitro and In Vivo Study
    Moura, Victor J. G.
    Alencar, Allan K. N.
    Calasans-Maia, Jorge de Albuquerque
    da Silva, Jaqueline Soares
    Fraga, Carlos A. M.
    Zapata-Sudo, Gisele
    Barreiro, Eliezer J.
    Sudo, Roberto Takashi
    UROLOGY, 2015, 85 (05) : 1214.e17 - 1214.e21
  • [47] In vitro and in vivo metabolism of a novel cannabinoid-1 receptor inverse agonist, taranabant, in rats and monkeys
    Reddy, V. B. G.
    Doss, G. A.
    Karanam, B. V.
    Samuel, K.
    Lanza, T. J., Jr.
    Lin, L. S.
    Yu, N. X.
    Zhang, A. S.
    Raab, C. E.
    Stearns, R. A.
    Kumar, S.
    XENOBIOTICA, 2010, 40 (09) : 650 - 662
  • [48] Characterization of the in vivo and in vitro electrophysiological effects of the novel antiarrhythmic agent AZD7009 in atrial and ventricular tissue of the dog
    Carlsson, L
    Chartier, D
    Nattel, S
    JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 2006, 47 (01) : 123 - 132
  • [49] JN403, in vitro characterization of a novel nicotinic acetylcholine receptor α7 selective agonist
    Feuerbach, Dominik
    Nozulak, Joachim
    Lingenhoehl, Kurt
    McAllister, Kevin
    Hoyer, Daniel
    NEUROSCIENCE LETTERS, 2007, 416 (01) : 61 - 65
  • [50] In vitro and in vivo characterization of a novel long-acting GLP-1 receptor agonist, exendin-4-Fc fusion protein
    Lu, Lian
    Su, Xiaoqing
    Wang, Yantai
    Luo, Yi
    Yang, Jun
    Xie, Li
    Gao, Xuefeng
    Ma, Yaru
    Tian, Yaomei
    Yuan, Fengjiao
    He, Gu
    Zhou, Bailing
    Fan, Yingzi
    Zhang, Xueyan
    Huang, Rong
    Lam, Ying Ka
    Jiang, Lin
    Dai, Hua
    Zhao, Qian
    Liao, Xiaoyang
    Yang, Li
    RSC ADVANCES, 2017, 7 (85) : 54178 - 54187
12345