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- [21] Allosteric inhibition of SHP2 variants containing cancer-associated activating mutationsCANCER RESEARCH, 2018, 78 (13)Wildes, David论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAAay, Naing论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USABuckl, Andreas论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAHsieh, Daphne论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAJogalekar, Ashutosh S.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAKiss, Gert论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAKoltun, Elena S.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAMarquez, Abby论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAMellem, Kevin T.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USARomero, Jason论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USASaldajeno-Concar, Mae论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USASchulze, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USASemko, Chris M.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAWon, Walter论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USANichols, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAStahlhut, Carlos论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USATzitzilonis, Christos论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USAGill, Adrian L.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USASmith, Jacqueline A.论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Redwood City, CA USA Revolut Med, Redwood City, CA USA
- [22] Allosteric inhibition of SHP2 phosphatase inhibits cancers driven by receptor tyrosine kinasesNATURE, 2016, 535 (7610) : 148 - +Chen, Ying-Nan P.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USALaMarche, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAChan, Ho Man论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAFekkes, Peter论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAGarcia-Fortanet, Jorge论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAAcker, Michael G.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAAntonakos, Brandon论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAChen, Christine Hiu-Tung论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAChen, Zhouliang论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USACooke, Vesselina G.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USADobson, Jason R.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USADeng, Zhan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAFei, Feng论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAFirestone, Brant论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAFodor, Michelle论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAFridrich, Cary论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAGao, Hui论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAGrunenfelder, Denise论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAHao, Huai-Xiang论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAJacob, Jaison论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAHo, Samuel论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAHsiao, Kathy论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAKang, Zhao B.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAKarki, Rajesh论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAKato, Mitsunori论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USALarrow, Jay论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USALa Bonte, Laura R.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USALenoir, Francois论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USALiu, Gang论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USALiu, Shumei论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAMajumdar, Dyuti论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAMeyer, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAPalermo, Mark论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAPerez, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAPu, Minying论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAPrice, Edmund论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAQuinn, Christopher论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAShakya, Subarna论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAShultz, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USASlisz, Joanna论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAVenkatesan, Kavitha论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAWang, Ping论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAWarmuth, Markus论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAWilliams, Sarah论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAYang, Guizhi论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAYuan, Jing论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAZhang, Ji-Hu论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAZhu, Ping论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USARamsey, Timothy论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USAKeen, Nicholas J.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, 250 Massachusetts Ave, Cambridge, MA 02139 USA
- [23] Structural reorganization of SHP2 by oncogenic mutations and implications for oncoprotein resistance to allosteric inhibitionNature Communications, 9Jonathan R. LaRochelle论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyMichelle Fodor论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyVidyasiri Vemulapalli论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyMorvarid Mohseni论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyPing Wang论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyTravis Stams论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyMatthew J. LaMarche论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyRajiv Chopra论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyMichael G. Acker论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular PharmacologyStephen C. Blacklow论文数: 0 引用数: 0 h-index: 0机构: Harvard Medical School,Department of Biological Chemistry & Molecular Pharmacology
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- [25] Thermodynamic and Kinetic Destabilization of Triosephosphate Isomerase Resulting from the Mutation of Conserved and Non-conserved CysteinesPROTEIN AND PEPTIDE LETTERS, 2011, 18 (12): : 1290 - 1298Eugenia Cruces-Angeles, Ma论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, Mexico Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, MexicoCabrera, Nallely论文数: 0 引用数: 0 h-index: 0机构: Univ Nacl Autonoma Mexico, Inst Fisiol Celular, Dept Bioquim & Biol Estruct, Coyoacan 04510, DF, Mexico Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, MexicoPerez-Montfort, Ruy论文数: 0 引用数: 0 h-index: 0机构: Univ Nacl Autonoma Mexico, Inst Fisiol Celular, Dept Bioquim & Biol Estruct, Coyoacan 04510, DF, Mexico Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, MexicoReyes-Lopez, Cesar A.论文数: 0 引用数: 0 h-index: 0机构: Inst Politecn Nacl, ENMyH, Postgrad Inst Biomed Mol, Lab Invest Bioquim, Gustavo A Madero 07320, DF, Mexico Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, MexicoHernandez-Arana, Andres论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, Mexico Univ Autonoma Metropolitana Iztapalapa, Dept Quim, Area Biofis Quim, Iztapalapa 09340, DF, Mexico
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Novartis Pharmaceut, Global Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USADeng, Zhan论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, Ctr Prote Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Pharmaceut, Global Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USAFirestone, Brant论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, Oncol Dis Area, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Pharmaceut, Global Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USAFekkes, Peter论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, Ctr Prote Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Pharmaceut, Global Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USAFodor, Michelle论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, Ctr Prote Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Pharmaceut, Global Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USAFortin, Pascal D.论文数: 0 引用数: 0 h-index: 0机构: 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Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Global Discovery Chem, 250 Massachusetts Ave, Cambridge, MA 02139 USA
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