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- [1] Allosteric inhibition of SHP2 phosphataseABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253Fortanet, Jorge Garcia论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAChen, Christine论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAChen, Yingnan论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAChen, Zhouliang论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USADeng, Zhan论文数: 0 引用数: 0 h-index: 0机构: Novartis, Winchester, MA USA Novartis, Reading, MA USAFirestone, Brant论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAFekkes, Peter论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAFodor, Michelle论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAFortin, Pascal论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAFridrich, Cary论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAGrunenfelder, Denise论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAHo, Samuel论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAKang, Zhao论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAKarki, Rajesh论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAKato, Mitsunori论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis Inst BioMed Res, Comp Aided Drug Discovery, Cambridge, MA USA Novartis, Reading, MA USAKeen, Nick论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALabonte, Laura论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALarrow, Jay论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALenoir, Francois论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALiu, Gang论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALiu, Shumei论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALombardo, Franco论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAMajumdar, Dyuti论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAMeyer, Matthew论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAPalermo, Mark论文数: 0 引用数: 0 h-index: 0机构: Novartis, Rindge, MA USA Novartis, Reading, MA USAPerez, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAPu, Minying论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USARamsey, Timothy论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USASellers, William论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAShultz, Michael论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res Inc, Cambridge, MA USA Novartis, Reading, MA USAStams, Travis论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USATowler, Chris论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAWang, Ping论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAWilliams, Sarah论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USAZhang, Ji-Hu论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USALaMarche, Matthew论文数: 0 引用数: 0 h-index: 0机构: Novartis, Reading, MA USA Novartis, Reading, MA USA
- [2] Dual Allosteric Inhibition of SHP2 PhosphataseACS CHEMICAL BIOLOGY, 2018, 13 (03) : 647 - 656Fodor, Michelle论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAPrice, Edmund论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAWang, Ping论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALu, Hengyu论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAArgintaru, Andreea论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAChen, Zhouliang论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAGlick, Meir论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAHao, Huai-Xiang论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAKato, Mitsunori论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAKoenig, Robert论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALaRochelle, Jonathan R.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALiu, Gang论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAMcNeill, Eric论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAMajumdar, Dyuti论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USANishiguchi, Gisele A.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAPerez, Lawrence B.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAParis, Gregory论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAQuinn, Christopher M.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USARamsey, Timothy论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USASendzik, Martin论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAShultz, Michael David论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAWilliams, Sarah L.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAStams, Travis论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USABlacklow, Stephen C.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USAAcker, Michael G.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USALaMarche, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Cambridge, MA 02139 USA
- [3] Destabilization of the SHP2 and SHP1 protein tyrosine phosphatase domains by a non-conserved "backdoor" cysteineBIOCHEMISTRY AND BIOPHYSICS REPORTS, 2022, 32Yarnall, Matthew T. N.论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USAKim, Sean H.论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USAKorntner, Samuel论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USABishop, Anthony C.论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USA
- [4] Targeting a Cryptic Allosteric Site for Selective Inhibition of the Oncogenic Protein Tyrosine Phosphatase Shp2BIOCHEMISTRY, 2015, 54 (02) : 497 - 504Chio, Cynthia M.论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USALim, Christopher S.论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USABishop, Anthony C.论文数: 0 引用数: 0 h-index: 0机构: Amherst Coll, Dept Chem, Amherst, MA 01002 USA Amherst Coll, Dept Chem, Amherst, MA 01002 USA
- [5] Identifying a non-conserved site for achieving allosteric covalent inhibition of CECR2ACTA PHARMACOLOGICA SINICA, 2025,Tang, Cai-ling论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaLi, Yuan-qing论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaDu, Xi-kun论文数: 0 引用数: 0 h-index: 0机构: Soochow Univ, Suzhou Med Coll, Sch Life Sci, Ctr Syst Biol,Dept Bioinformat, Suzhou 215123, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaFang, Xiao-xia论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaGuang, Yi-man论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaLi, Pei-zhuo论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaChen, Shuang论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaXue, Sheng-yu论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaYu, Jia-min论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaLiu, Xiao-yi论文数: 0 引用数: 0 h-index: 0机构: Soochow Univ, Suzhou Med Coll, Sch Life Sci, Ctr Syst Biol,Dept Bioinformat, Suzhou 215123, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaLuo, Yi-pan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Zunyi Med Univ, Sch Pharm, Zunyi 563000, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaZhou, Lan-xin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Guizhou Med Univ, Sch Pharm, Guiyang 550004, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaLuo, Cheng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Guizhou Med Univ, Sch Pharm, Guiyang 550004, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaXiong, Huan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaLiang, Zhong-jie论文数: 0 引用数: 0 h-index: 0机构: Soochow Univ, Suzhou Med Coll, Sch Life Sci, Ctr Syst Biol,Dept Bioinformat, Suzhou 215123, Peoples R China Soochow Univ, Jiangsu Prov Engn Res Ctr Precis Diagnost & Therap, Suzhou 215123, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaDing, Hong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China Guizhou Med Univ, Sch Pharm, Guiyang 550004, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China
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