Synthesis of both enantiomers of alpha-(trifluoromethyl)butyrine and alpha-(trifluoromethyl)phenylalanine

被引：0
|
作者：
Bravo, P
Viani, F
Zanda, M
Kukhar, VP
Soloshonok, VA
Fokina, N
Shishkin, OV
Struchkov, YT
机构：
[1] UKRAINIAN ACAD SCI, INST BIOORGAN CHEM & PETROCHEM, UA-253660 KIEV, UKRAINE
[2] RUSSIAN ACAD SCI, AU NESMEYANOV INST ORGANOELEMENT CPDS, MOSCOW, RUSSIA
来源：
GAZZETTA CHIMICA ITALIANA | 1996年 / 126卷 / 10期
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
The synthesis of both enantiomers of alpha-(trinuoromethyl)butyrine and alpha-(trifluoromethyl)phenylalanine was accomplished by desulfurization and deprotection of the beta-trifluoromethyl sulfoxides, obtained in the condensation of the corresponding optically pure alkyl p-tolyl sulfoxides with N-alkoxycarbonylimines of methyl 3,3,3-trifluoropyruvate.
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收藏
页码：645 / 652
页数：8
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