Microwave-assisted cross-coupling of 3-chloro-2-pyrazolines and 3-chloro-1-phenyl-1,4,5,6-tetrahydropyridazine with aryl boronic acids

被引：18
|
作者：
Wang, HJ
Keilman, J
Pabba, C
Chen, ZJ
Gregg, BT
机构：
[1] Albany Mol Res Inc, Botell Res Ctr, Bothell, WA 98011 USA
[2] Albany Mol Res Inc, Dept Combinatorial Parallel Synth, Albany, NY 12212 USA
来源：
TETRAHEDRON LETTERS | 2005年 / 46卷 / 15期
关键词：
2-pyrazoline; 1,4,5,6-tetrahydropyridazine; palladium; cross-coupling; boronic acids; microwave irradiation;
D O I：
10.1016/j.tetlet.2005.02.075
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
3-Chloro-l-phenyl-2-pyrazoliiie and 3-chloo-1-phenyl-1,4,5,6-tetrahydropyridazine were coupled with aryl boronic acids in good yields under microwave heating conditions (140 degrees C, 5 min). (c) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码：2631 / 2634
页数：4
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