New, efficient, selective, and one-pot method for acylation of amines

被引:7
|
作者
Basanagouda, Mahantesha [1 ]
Kulkarni, Manohar V. [1 ]
Kalkhambkar, Raj G. [2 ]
Kulkarni, Geeta M. [2 ]
机构
[1] Karnatak Univ, Dept Chem, Dharwad 580003, Karnataka, India
[2] Karnatak Sci Coll, Dept Chem, Dharwad, Karnataka, India
关键词
acetic acid; acetylation; amines; hydrazine hydrate; propionic acid; propionylation;
D O I
10.1080/00397910801997538
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Hydrazine hydrate with acetic and propionic acids was an efficient reagent for acylation of primary and secondary amines at reflux temperatures. The reported one-pot method is high-yielding, simple, mild, and inexpensive.
引用
收藏
页码:2929 / 2940
页数:12
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