Pictet-Spengler synthesis of some thiophene[c]-fused β-carbolines

被引：3
|
作者：
Abu Safieh, Kayed A. [2 ]
Moosa, Basem A. [3 ]
El-Abadelah, Mustafa M. [3 ]
Sabri, Salim S. [4 ]
Voelter, Wolfgang [1 ]
机构：
[1] Univ Tubingen, Interfak Inst Biochem, Tubingen, Germany
[2] Hashemite Univ, Fac Sci, Dept Chem, Zarqa, Jordan
[3] Univ Jordan, Fac Sci, Dept Chem, Amman, Jordan
[4] Univ Sharjah, Shajah, U Arab Emirates
来源：
MONATSHEFTE FUR CHEMIE | 2008年 / 139卷 / 02期
关键词：
3-(3-aminothien-2-yl)indole; Pictet-Spengler reaction; thieno[2,3-c]-beta-carbolines;
D O I：
10.1007/s00706-007-0763-6
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
5-(Substituted) thieno[2',3':5,6]pyrido[3,4-b]indoles were synthesized via cyclocondensation of 3-(3-aminothien-2-yl)indole with the appropriate aldehyde in the presence of boron trifluoride etherate under Pictet-Spengler reaction conditions. The constitution of the new compounds is evidenced from analytical and spectral (NMR and MS) data.
引用
收藏
页码：147 / 151
页数：5
相关论文
共 50 条
  • [1] Pictet-Spengler Synthesis of Some Thiophene[c]-Fused β-Carbolines
    Kayed A. Abu Safieh
    Basem A. Moosa
    Mustafa M. El-Abadelah
    Salim S. Sabri
    Wolfgang Voelter
    [J]. Monatshefte für Chemie - Chemical Monthly, 2008, 139 : 147 - 151
  • [2] Pictet-Spengler synthesis of pyrazole-fused β-carbolines
    Fasfous, II
    El-Abadelah, MM
    Sabri, SS
    [J]. JOURNAL OF HETEROCYCLIC CHEMISTRY, 2002, 39 (01) : 225 - 227
  • [3] The Chiral Pool in the Pictet-Spengler Reaction for the Synthesis of β-Carbolines
    Dalpozzo, Renato
    [J]. MOLECULES, 2016, 21 (06)
  • [4] Pictet-Spengler Synthesis of Perfluoroalkylated Tetrahydro-γ-carbolines and Tetrahydropyrrolopyrazines
    Voznesenskaia, Natalia G.
    Shmatova, Olga I.
    Nenajdenko, Valentine G.
    [J]. SYNTHESIS-STUTTGART, 2020, 52 (02): : 263 - 272
  • [5] Synthesis of tetrahydro-β-carbolines and studies of the Pictet-Spengler reaction
    Ducrot, P
    Rabhi, C
    Thal, C
    [J]. TETRAHEDRON, 2000, 56 (17) : 2683 - 2692
  • [6] Pictet-Spengler synthesis of tetrahydro-β-carbolines using vinylsulfonylmethyl resin
    Connors, RV
    Zhang, AJ
    Shuttleworth, SJ
    [J]. TETRAHEDRON LETTERS, 2002, 43 (37) : 6661 - 6663
  • [7] Stereoselective Synthesis of Functionalized Tetrahydro-β-Carbolines via Pictet-Spengler Reaction
    Vavsari, Vaezeh Fathi
    Dianati, Vahid
    Ramezanpour, Sorour
    Balalaie, Saeed
    [J]. SYNLETT, 2015, 26 (14) : 1955 - 1960
  • [8] Water as an efficient medium for the synthesis of tetrahydro-β-carbolines via Pictet-Spengler reactions
    Saha, Biswajit
    Sharma, Sunil
    Sawant, Devesh
    Kundu, Bijoy
    [J]. TETRAHEDRON LETTERS, 2007, 48 (08) : 1379 - 1383
  • [9] Synthesis of Tetrahydro-β-carbolines by a Manganese-Catalysed Oxidative Pictet-Spengler Reaction
    Shao, Zhihui
    Zhang, Xiaoyu
    Li, Xinyan
    Wang, Weilin
    Ding, Jiaqiao
    Cui, Bing
    Zhao, Mingqin
    [J]. CHEMISTRY-A EUROPEAN JOURNAL, 2023, 29 (39)
  • [10] Pictet-Spengler Synthesis of Quinoline-Fused Porphyrins and Phenanthroline-Fused Diporphyrins
    Gao, Ke
    Fukui, Norihito
    Jung, Seok Ii
    Yorimitsu, Hideki
    Kim, Dongho
    Osuka, Atsuhiro
    [J]. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2016, 55 (42) : 13038 - 13042
12345