The Design and Synthesis of Pyrolle-Carbaldehydes as HIV-1 Integrase Strand-Transfer Inhibitors

被引：0
|
作者：
Hewer, Raymond [1 ]
Traut, Telisha [1 ,2 ]
Williams, Bradley [2 ]
Coates, Judy [1 ]
机构：
[1] MINTEK, Johannesburg, South Africa
[2] Univ Johannesburg, Johannesburg, South Africa
来源：
ANTIVIRAL RESEARCH | 2011年 / 90卷 / 02期
关键词：
D O I：
10.1016/j.antiviral.2011.03.087
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
101
引用
收藏
页码：A50 / A50
页数：1
相关论文
共 50 条
  • [11] More pressure on integrase strand-transfer inhibitors?
    Pozniak, Anton L.
    Venter, W. D. Francois
    LANCET HIV, 2023, 11 (05): : e278 - e280
  • [12] Transmitted resistance to HIV integrase strand-transfer inhibitors: right on schedule
    Hurt, Christopher B.
    ANTIVIRAL THERAPY, 2011, 16 (02) : 137 - 140
  • [13] Prevalence of resistance to integrase strand-transfer inhibitors (INSTIs) among untreated HIV-1 infected patients in Morocco
    Alaoui N.
    El Alaoui M.A.
    Touil N.
    El Annaz H.
    Melloul M.
    Tagajdid R.
    Hjira N.
    Boui M.
    El Fahime E.M.
    Mrani S.
    BMC Research Notes, 11 (1)
  • [14] Integrase strand-transfer inhibitors for treatment of early HIV infection A case series
    Teira, Ramon
    Gutierrez, Mar
    Galindo, Pepa
    Martinez, Elisa
    Munoz, Pepa
    de la Fuente, Belen
    Tellez, Francisco
    Montero, Marta
    MEDICINE, 2019, 98 (35) : e16866
  • [15] Primary resistance to integrase strand-transfer inhibitors in Europe
    Casadella, M.
    van Ham, P. M.
    Noguera-Julian, M.
    van Kessel, A.
    Pou, C.
    Hofstra, L. M.
    Santos, J. R.
    Garcia, F.
    Struck, D.
    Alexiev, I.
    Kran, A. M. Bakken
    Hoepelman, A. I.
    Kostrikis, L. G.
    Somogyi, S.
    Liitsola, K.
    Linka, M.
    Nielsen, C.
    Otelea, D.
    Paraskevis, D.
    Poljak, M.
    Puchhammer-Stoeckl, E.
    Stanekova, D.
    Stanojevic, M.
    Van Laethem, K.
    Lepej, S. Zidovec
    Clotet, B.
    Boucher, C. A. B.
    Paredes, R.
    Wensing, A. M. J.
    JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 2015, 70 (10) : 2885 - 2888
  • [16] Chromone and chromanone derivatives as strand transfer inhibitors of HIV-1 integrase
    Park, Jang Hyun
    Lee, Seung Uk
    Kim, Sang Hoon
    Shin, Seo Yeong
    Lee, Jae Yeol
    Shin, Cha-Gyun
    Yoo, Kyung Ho
    Lee, Yong Sup
    ARCHIVES OF PHARMACAL RESEARCH, 2008, 31 (01) : 1 - 5
  • [17] Ruthenium arene complexes as HIV-1 integrase strand transfer inhibitors
    Carcelli, Mauro
    Bacchi, Alessia
    Pelagatti, Paolo
    Rispoli, Gabriele
    Rogolino, Dominga
    Sanchez, Tino W.
    Sechi, Mario
    Neamati, Nouri
    JOURNAL OF INORGANIC BIOCHEMISTRY, 2013, 118 : 74 - 82
  • [18] Chromone and chromanone derivatives as strand transfer inhibitors of HIV-1 integrase
    Jang Hyun Park
    Seung Uk Lee
    Sang Hoon Kim
    Seo Yeong Shin
    Jae Yeol Lee
    Cha-Gyun Shin
    Kyung Ho Yoo
    Yong Sup Lee
    Archives of Pharmacal Research, 2008, 31 : 1 - 5
  • [19] Inhibition of matrix metalloproteinases by HIV-1 integrase strand transfer inhibitors
    Foster, Emma G. G.
    Palermo, Nicholas Y. Y.
    Liu, Yutong
    Edagwa, Benson
    Gendelman, Howard E. E.
    Bade, Aditya N. N.
    FRONTIERS IN TOXICOLOGY, 2023, 5
  • [20] Lack of activity of HIV-1 integrase strand-transfer inhibitors on recombinase activating gene (RAG) activity at clinically relevant concentrations
    Demirdjian, Sally
    Duong, Vincent N.
    Byrum, Jennifer N.
    Nayak, Arabinda
    Mckinney, Cooper B.
    Perry, Jason K.
    Callebaut, Christian
    Rodgers, Karla K.
    Falkard, Brie
    Feng, Joy Y.
    MICROBIOLOGY SPECTRUM, 2025, 13 (01)
12345