Targeting Pyruvate Kinase M2 As a Novel Therapeutic Strategy Against Liver Fibrosis and Hepatocellular Carcinoma

被引:0
|
作者
Zheng, Dandan [1 ]
Lin, Zelong [1 ,2 ]
Hu, Kaishun [3 ]
Lan, Tian [4 ]
Holmes, Jacinta A. [5 ,6 ,7 ]
Song, Zhenghui [2 ,8 ]
He, Lu [1 ]
Jiang, Yuchuan [1 ]
Chen, Peng [1 ,2 ]
Tu, Mengxian [1 ]
Chen, Hengxing [3 ]
Hu, Qiaoting [1 ]
Qu, Chen [1 ,2 ]
Lin, Wenyu [5 ,6 ,7 ]
Li, Aimin [2 ,8 ]
Chung, Raymond T. [5 ,6 ,7 ]
Hong, Jian [1 ,2 ]
机构
[1] Southern Med Univ, Integrated Hosp Tradit Chinese Med, Dept Abdominal Surg, Guangzhou, Guangdong, Peoples R China
[2] Southern Med Univ, Canc Ctr, Guangzhou, Guangdong, Peoples R China
[3] Sun Yat Sen Univ, Sun Yat Sen Mem Hosp, Guangzhou, Guangdong, Peoples R China
[4] Guangdong Pharmaceut Univ, Guangzhou, Guangdong, Peoples R China
[5] Massachusetts Gen Hosp, Liver Ctr, Boston, MA 02114 USA
[6] Massachusetts Gen Hosp, Gastrointestinal Div, Boston, MA 02114 USA
[7] Harvard Med Sch, Boston, MA USA
[8] Southern Med Univ, Integrated Hosp Tradit Chinese Med, Dept Hepatol, Guangzhou, Guangdong, Peoples R China
关键词
D O I
暂无
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
1120
引用
收藏
页码:646A / 647A
页数:2
相关论文
共 50 条
  • [21] Pyruvate kinase M2 at a glance
    Yang, Weiwei
    Lu, Zhimin
    JOURNAL OF CELL SCIENCE, 2015, 128 (09) : 1655 - 1660
  • [22] Prospects for immunotherapy as a novel therapeutic strategy against hepatocellular carcinoma
    Yu Akazawa
    Toshihiro Suzuki
    Toshiaki Yoshikawa
    Shoichi Mizuno
    Yasunari Nakamoto
    Tetsuya Nakatsura
    World Journal of Meta-Analysis, 2019, 7 (03) : 80 - 95
  • [23] Selective Covalent Targeting of Pyruvate Kinase M2 Using Arsenous Warheads
    Wang, Jingyao
    Zhou, Shaoqing
    Cheng, Yan
    Cheng, Lin
    Qin, Ying
    Zhang, Zhenfeng
    Bi, Aiwei
    Xiang, Huaijiang
    He, Xinheng
    Tian, Xiaoxu
    Liu, Wenbin
    Zhang, Jian
    Peng, Chao
    Zhu, Zhengjiang
    Huang, Min
    Li, Ying
    Zhuang, Guanglei
    Tan, Li
    JOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (04) : 2608 - 2621
  • [24] Search progress of pyruvate kinase M2 (PKM2) in organ fibrosis
    Lv, Shumei
    Cao, Mengfei
    Luo, Jie
    Fu, Kewei
    Yuan, Wei
    MOLECULAR BIOLOGY REPORTS, 2024, 51 (01)
  • [25] Lapachol inhibits glycolysis in cancer cells by targeting pyruvate kinase M2
    Babu, Mani Shankar
    Mahanta, Sailendra
    Lakhter, Alexander J.
    Hato, Takashi
    Paul, Subhankar
    Naidu, Samisubbu R.
    PLOS ONE, 2018, 13 (02):
  • [26] SH2 domain-containing phosphatase 1 regulates pyruvate kinase M2 in hepatocellular carcinoma
    Tai, Wei-Tien
    Hung, Man-Hsin
    Chu, Pei-Yi
    Chen, Yao-Li
    Chen, Li-Ju
    Tsai, Ming-Hsien
    Chen, Min-Husan
    Shiau, Chung-Wai
    Boo, Yin-Pin
    Chen, Kuen-Feng
    ONCOTARGET, 2016, 7 (16) : 22193 - 22205
  • [27] Targeting Pyruvate Kinase M2 Phosphorylation Reverses Aggressive Cancer Phenotypes
    Apostolidi, Maria
    Vathiotis, Ioannis A.
    Muthusamy, Viswanathan
    Gaule, Patricia
    Gassaway, Brandon M.
    Rimm, David L.
    Rinehart, Jesse
    CANCER RESEARCH, 2021, 81 (16) : 4346 - 4359
  • [28] Targeting of the glycolytic keyregulator pyruvate kinase subtype M2 by peptide aptamers
    Spoden, G
    Mazurek, S
    Morandell, D
    Eigenbrodt, E
    Zwerschke, W
    INTERNATIONAL JOURNAL OF OBESITY, 2005, 29 : S5 - S5
  • [29] Targeting RFX-1 as a novel therapeutic strategy in hepatocellular carcinoma
    Su, Jung-Chen
    CANCER RESEARCH, 2015, 75
  • [30] Pyruvate Kinase M2: A Novel Regulator of Brown and Fat Adipogenesis
    Knoxville, Presley Dowker
    OBESITY, 2021, 29 : 149 - 149