An efficient one-pot, purification-free, preparation of amides using polymer-supported reagents

被引：15

作者：

Lannuzel, M ^{[1
]}

Lamothe, M ^{[1
]}

Perez, M ^{[1
]}

机构：

[1] Ctr Rech Pierre Fabre, F-81106 Castres 06, France

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 38期

关键词：

D O I：

10.1016/S0040-4039(01)01387-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new one-pot method for amide preparation using polymer-supported carbodiimide is reported. It incorporated the use of HOBT to improve the reactivity of the supported reagent and expand the scope of this reaction. HOBT could then be subsequently easily removed from the medium with a supported carbonate base. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

页码：6703 / 6705

页数：3

共 50 条

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