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- [1] Potent and selective pyridone BTK inhibitors with an induced fit binding mode and activity vs. mutant forms of BTK[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Crawford, James J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USAJohnson, Adam论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Biochem Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USAWei, BinQing论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Computat Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USAOrtwine, Daniel F.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Computat Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USAKohli, Pawan Bir论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Biochem Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USAYoung, Wendy B.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA
- [2] Optimization of a novel piperazinone series as potent selective peripheral covalent BTK inhibitors[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 60Ma, Bin论文数: 0 引用数: 0 h-index: 0机构: Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAMetrick, Claire M.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Biophys, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAGu, Chungang论文数: 0 引用数: 0 h-index: 0机构: Biogen, Drug Metab & Pharmacokinet, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAHoemberger, Marc论文数: 0 引用数: 0 h-index: 0机构: Biogen, Bioassays & High Throughput Screens, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USABajrami, Bekim论文数: 0 引用数: 0 h-index: 0机构: Biogen, Chem Biol & Prote, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USABame, Eris论文数: 0 引用数: 0 h-index: 0机构: Biogen, Translat Sci, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAHuang, Jiansheng论文数: 0 引用数: 0 h-index: 0机构: Biogen, Drug Metab & Pharmacokinet, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAMingueneau, Michael论文数: 0 引用数: 0 h-index: 0机构: Biogen, Multiple Sclerosis & Neurorepair Res, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAMurugan, Paramasivam论文数: 0 引用数: 0 h-index: 0机构: Biogen, Bioassays & High Throughput Screens, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USASantoro, Joseph C.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Bioassays & High Throughput Screens, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USATang, Hao论文数: 0 引用数: 0 h-index: 0机构: Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAWang, Ti论文数: 0 引用数: 0 h-index: 0机构: Biogen, Bioassays & High Throughput Screens, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USAHopkins, Brian T.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USA Biogen, Med Chem, 225 Binney St, Cambridge, MA 02142 USA
- [3] Purine derivatives as potent BTK inhibitors for autoimmune diseases[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242Shi, Qing论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USALiu, Chunjian论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USALin, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USADyckman, Alaric J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USALi, Hedy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAVandevier, Lauren E.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USACavallaro, Cullen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USASpergel, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USABurke, James R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USATebben, Andrew论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAStrnad, Joann论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USASurti, Neha论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAMuckelbauer, Jodi K.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAMcintyre, Kim论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USALeftheris, Katerina论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USACarter, Percy H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USATino, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USADelucca, George V.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USA
- [4] REDX08608, a Novel, Potent and Selective, Reversible BTK Inhibitor with Efficacy and Equivalent Potency Against Wild-Type and Mutant C481S BTK[J]. BLOOD, 2016, 128 (22)Guisot, Nicolas E. S.论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandBest, Stuart A.论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandWright, Victoria论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandThomason, Andrew论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandWoyach, Jennifer A.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Hematol, Dept Internal Med, Columbus, OH USA Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandMantel, Rose论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Div Hematol, Dept Internal Med, Columbus, OH USA Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandMcClanahan, Fabienne论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Ctr Comprehens Canc, Columbus, OH USA Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandAbet, Valentina论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandCastagna, Diana论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandCousin, Peggy论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandEmmerich, Juliette论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandHo, Kelvin论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandKelly, James Russell论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandKing-Tours, James论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandLyons, Kristina论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandMuller, Melanie论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandRefuerzo, Julienne论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandSargent, Louise论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandTalab, Fatima论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandBingham, Matilda论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandPhillips, Caroline论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, EnglandArmer, Richard论文数: 0 引用数: 0 h-index: 0机构: Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England Redx Oncol Ltd, Redx Pharma Plc, Alderley Edge, England
- [5] Discovery of pyrazolopyrimidine derivatives as potent BTK inhibitors with effective anticancer activity in MCL[J]. BIOORGANIC CHEMISTRY, 2019, 89Ran, Fansheng论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaLiu, Yang论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Lymphoma & Myeloma, Houston, TX 77030 USA Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaLiu, Meixia论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaZhang, Daoguang论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaWang, Peng论文数: 0 引用数: 0 h-index: 0机构: Shandong Qidu Pharmaceut Co Ltd, 28 Renmin East Rd, Zibo 255400, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaDong, Junze论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaTang, Wendi论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R ChinaZhao, Guisen论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China Shandong Univ, Sch Pharmaceut Sci, Minist Educ, Dept Med Chem,Key Lab Chem Biol, 44 West Culture Rd, Jinan 250012, Shandong, Peoples R China
- [6] Nicotinamide derivatives as potent BTK inhibitors for autoimmune diseases[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242De Lucca, George V.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USAShi, Qing论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USALiu, Chunjian论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USATebben, Andrew论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USAStrnad, Joann论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USASurti, Neha论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USAMuckelbauer, Jodi K.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USAMcintyre, Kim论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USABurke, James R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USALeftheris, Katerina论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USACarter, Percy H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USATino, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USAChang, Chiehying论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08540 USA
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