Biological characterization of TAS3681, a new type of androgen receptor antagonist with androgen receptor downregulating activity

被引:0
|
作者
Minamiguchi, K. [1 ]
Seki, M. [1 ]
Aoyagi, H. [1 ]
Mori, T. [1 ]
Kajiwara, D. [1 ]
Masuko, N. [1 ]
Fujita, R. [1 ]
Okajima, S. [1 ]
Hayashi, Y. [1 ]
Sasaki, E. [1 ]
Utsugi, T. [1 ]
机构
[1] Taiho Pharmaceut Co Ltd, Tsukuba Res Ctr, Ibaraki, Japan
关键词
D O I
10.1016/S0959-8049(14)70441-1
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
315
引用
收藏
页码:103 / 103
页数:1
相关论文
共 50 条
  • [31] The impact of androgen-induced translation in modulating androgen receptor activity
    Israel, Justus S.
    Marcelin, Laura-Maria
    Mehralivand, Sherif
    Scholze, Jana
    Hofmann, Joerg
    Stope, Matthias B.
    Puhr, Martin
    Thomas, Christian
    Erb, Holger H. H.
    BIOLOGY DIRECT, 2024, 19 (01)
  • [32] ABSENCE OF ANDROGEN RECEPTOR AFFINITY FOR MK-208, A NEW H-2-RECEPTOR ANTAGONIST
    LIANG, T
    CLINICAL RESEARCH, 1984, 32 (02): : A283 - A283
  • [33] Androgen-receptor coregulators mediate the suppressive effect of androgen signals on vitamin D receptor activity
    Ting, HJ
    Bao, BY
    Hsu, CL
    Lee, YF
    ENDOCRINE, 2005, 26 (01) : 1 - 9
  • [34] Androgen-receptor coregulators mediate the suppressive effect of androgen signals on vitamin D receptor activity
    Huei-Ju Ting
    Bo-Ying Bao
    Cheng-Lung Hsu
    Yi-Fen Lee
    Endocrine, 2005, 26 : 1 - 9
  • [35] Catalytic cleavage of the androgen receptor messenger RNA and functional inhibition of androgen receptor activity by a hammerhead ribozyme
    Chen, S
    Song, CS
    Lavrovsky, Y
    Bi, BY
    Vellanoweth, R
    Chatterjee, B
    Roy, AK
    MOLECULAR ENDOCRINOLOGY, 1998, 12 (10) : 1558 - 1566
  • [36] Regulation of androgen receptor activity by the nuclear receptor corepressor SMRT
    Liao, GQ
    Chen, LY
    Zhang, AH
    Godavarthy, A
    Xia, F
    Ghosh, JC
    Li, H
    Chen, JD
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2003, 278 (07) : 5052 - 5061
  • [37] MODULATION OF ANDROGEN RECEPTOR TRANSCRIPTIONAL ACTIVITY BY THE ESTROGEN-RECEPTOR
    KUMAR, MV
    LEO, ME
    TINDALL, DJ
    JOURNAL OF ANDROLOGY, 1994, 15 (06): : 534 - 542
  • [38] Androgen action on hepatic vitellogenin synthesis in the eel, Anguilla japonica is suppressed by an androgen receptor antagonist
    Kwon, HC
    Choi, SH
    Kim, YU
    Son, SO
    Kwon, JY
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 2005, 96 (02): : 175 - 178
  • [39] Design, synthesis, and biological characterization of metabolically stable selective androgen receptor modulators
    Marhefka, CA
    Gao, WQ
    Chung, KW
    Kim, JY
    He, YL
    Yin, DH
    Bohl, C
    Dalton, JT
    Miller, DD
    JOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (04) : 993 - 998
  • [40] Discovery and biological evaluation of novel androgen receptor antagonist for castration-resistant prostate cancer
    Yu, Jiang
    Zhang, Lanxi
    Yan, Guoyi
    Zhou, Peiting
    Cao, Chaoguo
    Zhou, Fei
    Li, Xinghai
    Chen, Yuanwei
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 171 : 265 - 281