Solvent-free copper-catalyzed N-arylation of amino alcohols and diamines with aryl halides

被引：34
|
作者：
Yin, Huiqing [1 ]
Jin, Ming [1 ]
Chen, Wei [1 ]
Chen, Chen [1 ]
Zheng, Likang [1 ]
Wei, Ping [1 ]
Han, Shiqing [1 ,2 ]
机构：
[1] Nanjing Univ Technol, Coll Biotechnol & Pharmaceut Engn, Nanjing 210009, Peoples R China
[2] Chinese Acad Sci, Key Lab Synthet Chem Nat Subst, Shanghai Inst Organ Chem, Shanghai 200032, Peoples R China
来源：
TETRAHEDRON LETTERS | 2012年 / 53卷 / 10期
基金：
中国国家自然科学基金;
关键词：
Copper-catalyzed; N-arylation; Solvent-free; Amino alcohols; Diamines; NITROGEN-CONTAINING HETEROCYCLES; C-N; BOND FORMATION; COUPLING REACTIONS; EFFICIENT; LIGAND; AMINATION; IODIDES; MILD; AMIDATION;
D O I：
10.1016/j.tetlet.2011.12.130
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A simple and mild method for the coupling of aryl halides with amino alcohols and diamines is described. The reactions can be performed under ligand-free and solvent-free conditions, and generate the products in good yield. (C) 2012 Elsevier Ltd. All rights reserved.
引用
收藏
页码：1265 / 1270
页数：6
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