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- [41] The discovery of 2-fluoro-N-(3-fluoro-4-(5-((4-morpholinobutyl)amino)-1,3,4-oxadiazol-2-yl)phenyl)benzamide, a full agonist of the alpha-7 nicotinic acetylcholine receptor showing efficacy in the novel object recognition model of cognition enhancementBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (10) : 3531 - 3534Skidmore, John论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandAtcha, Zeenat论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D China, Ctr Cognit & Neurodegenerat, Singapore 138667, Singapore GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandBoucherat, Emmanuelle论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandCastelletti, Laura论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D China, Ctr Cognit & Neurodegenerat, Singapore 138667, Singapore GlaxoSmithKline, Mol Discovery Res, I-37135 Verona, Italy GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandChen, Deborah W.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandCoppo, Frank T.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Mol Discovery Res, Collegeville, PA 19426 USA GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandCutler, Leanne论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandDunsdon, Rachel M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandHeath, Bronagh M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Safety Assessment, Ware SG12 0DP, Herts, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandHutchings, Rio论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandHurst, David N.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandJaved, Sahar论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandMartin, Samuel论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandMaskell, Emma S. L.论文数: 0 引用数: 0 h-index: 0机构: Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandNorton, David论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandPemberton, Darrel J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D China, Ctr Cognit & Neurodegenerat, Singapore 138667, Singapore GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandRedshaw, Sally论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandRutter, Richard论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D China, Ctr Cognit & Neurodegenerat, Singapore 138667, Singapore GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandSehmi, Sanjeet S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandScoccitti, Tiziana论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandTemple, Hannah E.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandTheobald, Pam论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandWard, Robert W.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, EnglandWilson, David M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Neurosci Ctr Excellence Drug Discovery, Harlow CM19 5AW, Essex, England
- [42] The potent and selective alpha 4 beta 2*/alpha 6*-nicotinic acetylcholine receptor partial agonist 2-[5-[5-((S)Azetidin-2-ylmethoxy) -3-pyridinyl]-3-isoxazolyl]ethanol demonstrates antidepressive-like behavior in animal models and a favorable ADME-tox profilePHARMACOLOGY RESEARCH & PERSPECTIVES, 2014, 2 (02):Yu, Li-Fang论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USA East China Normal Univ, Shanghai Engn Res Ctr Mol Therapeut & New Drug De, Inst Drug Design & Dev, Shanghai 200062, Peoples R China Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAEaton, J. Brek论文数: 0 引用数: 0 h-index: 0机构: Barrow Neurol Inst, Div Neurobiol, Phoenix, AZ 85013 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAZhang, Han-Kun论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USA East China Normal Univ, Inst Biomed Sci, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai 200241, Peoples R China Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USASabath, Emily论文数: 0 引用数: 0 h-index: 0机构: PsychoGenics Inc, Tarrytown, NY USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAHanania, Taleen论文数: 0 引用数: 0 h-index: 0机构: PsychoGenics Inc, Tarrytown, NY USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USALi, Guan-Nan论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAvan Breemen, Richard B.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAWhiteaker, Paul论文数: 0 引用数: 0 h-index: 0机构: Barrow Neurol Inst, Div Neurobiol, Phoenix, AZ 85013 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USALiu, Qiang论文数: 0 引用数: 0 h-index: 0机构: Barrow Neurol Inst, Div Neurobiol, Phoenix, AZ 85013 USA Barrow Neurol Inst, Div Neurol, Phoenix, AZ 85013 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAWu, Jie论文数: 0 引用数: 0 h-index: 0机构: Barrow Neurol Inst, Div Neurol, Phoenix, AZ 85013 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAChang, Yong-Chang论文数: 0 引用数: 0 h-index: 0机构: Barrow Neurol Inst, Div Neurobiol, Phoenix, AZ 85013 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USALukas, Ronald J.论文数: 0 引用数: 0 h-index: 0机构: Barrow Neurol Inst, Div Neurobiol, Phoenix, AZ 85013 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USABrunner, Dani论文数: 0 引用数: 0 h-index: 0机构: PsychoGenics Inc, Tarrytown, NY USA Columbia Univ, Dept Psychiat, NYSPI, New York, NY 10032 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USAKozikowski, Alan P.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USA Univ Illinois, Dept Med Chem & Pharmacognosy, 833 South Wood St, Chicago, IL 60612 USA