New growth hormone secretagogues:: C-terminal modified sulfonamide-analogues of NN703

被引：5
|
作者：
Peschke, B
Hansen, BS
机构：
[1] Novo Nordisk AS, Hlth Care Chem, DK-2760 Malov, Denmark
[2] Novo Nordisk AS, Diabet Biochem, DK-2880 Bagsvaerd, Denmark
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1999年 / 9卷 / 09期
关键词：
D O I：
10.1016/S0960-894X(99)00167-5
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
The C-terminal the orally active growth hormone secretagogue NN703 was changed to prepare analogues with inverse sulfonamides and inverse amides. The compounds showed high activity in a in vitro rat pituitary model. (C) 1999 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：1295 / 1298
页数：4
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