Synthesis of 5-aryl-1,2-dihydro-1-pyrrolizinones

被引:0
|
作者
Yu, H [1 ]
Wang, F [1 ]
Zhang, SF [1 ]
机构
[1] Shenyang Pharmaceut Univ, Shenyang 110015, Peoples R China
关键词
5-aryl-1,2-dihydro-1-pyrrolizinone; anti-inflammation; analgesic; synthesis;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
In order to search for new potent anti-inflammatory and analgesic agents in pyrrolizinones, the title compounds were designed and synthesized. A series of the compounds were prepared with two different synthetic schemes. Some of the compounds showed remarkable anti-inflammatory and/or analgesic activities on mice.
引用
收藏
页码:565 / 568
页数:4
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