Bifeprunox: a novel atypical antipsychotic sharing dopamine D(2,3,4) receptor and serotonin 5-HT(1A) receptor affinities

被引:0
|
作者
Marquis, K
Hertel, P
Reinders, JH
Van der Neut, M
Ronken, E
McCreary, AC
Herremans, AHJ
Hesselink, MB
机构
关键词
D O I
暂无
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:S487 / S487
页数:1
相关论文
共 50 条
  • [41] Involvement of dopamine (DA)/serotonin (5-HT)/sigma (σ) receptor modulation in mediating the antidepressant action of ropinirole hydrochloride, a D2/D3 doparnine receptor agonist
    Dhir, Ashish
    Kulkarni, S. K.
    BRAIN RESEARCH BULLETIN, 2007, 74 (1-3) : 58 - 65
  • [42] SELECTIVE 5-HT(1A)-RECEPTOR-MEDIATED AND 5-HT(2)-RECEPTOR-MEDIATED ADRENOCORTICOTROPIN RELEASE IN THE RAT - EFFECT OF REPEATED ANTIDEPRESSANT TREATMENTS
    GARTSIDE, SE
    ELLIS, PM
    SHARP, T
    COWEN, PJ
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1992, 221 (01) : 27 - 33
  • [43] Increase of 5-HT7 (serotonin-7) and 5-HT(1A) (serotonin-1A) receptor mRNA expression in rat hippocampus after adrenalectomy
    Le Corre S.
    Sharp T.
    Young A.H.
    Harrison P.J.
    Psychopharmacology, 1997, 130 (4) : 368 - 374
  • [44] Alterations in adolescent brain serotonin (5HT)1A, 5HT2A, and dopamine (D)2 receptor systems in a nonhuman primate model of early life adversity
    Wakeford, Alison G. P.
    Nye, Jonathon A.
    Morin, Elyse L.
    Mun, Jiyoung
    Meyer, Jerrold S.
    Goodman, Mark
    Howell, Leonard L.
    Sanchez, Mar M.
    NEUROPSYCHOPHARMACOLOGY, 2024, 49 (08) : 1227 - 1235
  • [45] Serotonin (5-HT)1A receptor agonism and 5-HT7 receptor antagonism ameliorate the subchronic phencyclidine-induced deficit in executive functioning in mice
    Rajagopal, Lakshmi
    Massey, Bill W.
    Michael, Eric
    Meltzer, Herbert Y.
    PSYCHOPHARMACOLOGY, 2016, 233 (04) : 649 - 660
  • [46] Atypical antipsychotic properties of blonanserin, a novel dopamine D2 and 5-HT2A antagonist
    Ohno, Yukihiro
    Okano, Motoki
    Imaki, Junta
    Tatara, Ayaka
    Okumura, Takahiro
    Shimizu, Saki
    PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 2010, 96 (02) : 175 - 180
  • [47] Serotonin (5-HT)1A receptor agonism and 5-HT7 receptor antagonism ameliorate the subchronic phencyclidine-induced deficit in executive functioning in mice
    Lakshmi Rajagopal
    Bill W. Massey
    Eric Michael
    Herbert Y. Meltzer
    Psychopharmacology, 2016, 233 : 649 - 660
  • [48] SEROTONIN 5-HT2A, DOPAMINE D2 AND NORADRENALINE ALPHA-1 ANTAGONISTS - ANALOGS OF THE ATYPICAL ANTIPSYCHOTIC SERTINDOLE
    ANDERSEN, K
    PERREGAARD, J
    LILJEFORS, T
    HYTTEL, J
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1995, 210 : 130 - MEDI
  • [49] Serotonin (5-HT) 5-HT2C receptor (5-HT2CR) positive allosteric modulators as novel neurotherapeutics
    Wild, Christopher
    McAllister, Carrie E.
    Wold, Eric A.
    Ding, Chunyong
    Anastasio, Noelle C.
    Fox, Robert G.
    Stutz, Sonja J.
    Chen, Haiying
    Tomlinson, Suzanne
    Cunningham, Kathryn
    Zhou, Jia
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251
  • [50] THE NOVEL 5-HT(1A)-RECEPTOR ANTAGONIST, SDZ 216-525, DECREASES 5-HT RELEASE IN RAT HIPPOCAMPUS IN-VIVO
    SHARP, T
    MCQUADE, R
    FOZARD, JR
    HOYER, D
    BRITISH JOURNAL OF PHARMACOLOGY, 1993, 109 (03) : 699 - 702