Acetylcholine binding protein-nicotinic receptor chimeras for delineating structure and determinants of ligand selectivity

被引:0
|
作者
Talley, Todd T. [1 ]
Nemecz, Akos [1 ]
Yamauchi, John G. [1 ]
Wu, Joshua [1 ]
Ho, Kwok-Yiu [1 ]
Sankaran, Banumathi [2 ]
Taylor, Palmer [1 ]
机构
[1] Univ Calif San Diego, Skaggs Sch Pharm & Pharmaceut Sci, La Jolla, CA 92093 USA
[2] Lawrence Berkeley Natl Lab, Berkeley Ctr Struct Biol, Berkeley, CA USA
关键词
D O I
10.1016/j.bcp.2011.07.018
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1028 / 1029
页数:2
相关论文
共 50 条
  • [31] Alpha-7 Nicotinic Acetylcholine Receptor (nAChR) Characteristics on the Acetylcholine Binding Protein
    Nemecz, Akos
    Taylor, Palmer
    FASEB JOURNAL, 2009, 23
  • [32] An allosteric binding site of the α7 nicotinic acetylcholine receptor revealed in a humanized acetylcholine-binding protein
    Delbart, Florian
    Brams, Marijke
    Gruss, Fabian
    Noppen, Sam
    Peigneur, Steve
    Boland, Sandro
    Chaltin, Patrick
    Brandao-Neto, Jose
    von Delft, Frank
    Touw, Wouter G.
    Joosten, Robbie P.
    Liekens, Sandra
    Tytgat, Jan
    Ulens, Chris
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 293 (07) : 2534 - 2545
  • [33] Characterization of Binding Site Interactions and Selectivity Principles in the α3β4 Nicotinic Acetylcholine Receptor
    Knox, Hailey J.
    Campello, Hugo Rego
    Lester, Henry A.
    Gallagher, Timothy
    Dougherty, Dennis A.
    JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 144 (35) : 16101 - 16117
  • [34] Investigating the ligand binding site of acetylcholine binding protein and the glycine receptor
    Yonkunas, Michael J.
    Liu, Zhenyu
    Speranskiy, Kirill
    Cascio, Mike
    Kurnikova, Maria
    BIOPHYSICAL JOURNAL, 2007, : 449A - 449A
  • [35] PROTEIN STRUCTURAL EFFECTS OF AGONIST BINDING TO THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    CASTRESANA, J
    FERNANDEZBALLESTER, G
    FERNANDEZ, AM
    LAYNEZ, JL
    ARRONDO, JLR
    FERRAGUT, JA
    GONZALEZROS, JM
    FEBS LETTERS, 1992, 314 (02) : 171 - 175
  • [37] Mapping the structure of the nicotinic acetylcholine receptor binding site by cysteine mutagenesis
    Hong, F
    Cohen, JB
    BIOPHYSICAL JOURNAL, 2001, 80 (01) : 462A - 463A
  • [38] PROTEIN-LIGAND INTERACTIONS - INTERACTION OF NITROSAMINES WITH NICOTINIC ACETYLCHOLINE-RECEPTOR
    KAPP, EA
    DAYA, S
    WHITELEY, CG
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1990, 167 (03) : 1383 - 1392
  • [39] Subunit interface selectivity of the α-neurotoxins for the nicotinic acetylcholine receptor
    Osaka, H
    Malany, S
    Kanter, JR
    Sine, SM
    Taylor, P
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1999, 274 (14) : 9581 - 9586