Isoxazolone Derivatives as Potent Inhibitors of PTP1B

被引：23
|
作者：
Kafle, Bhooshan [1 ]
Cho, Hyeongjin [1 ]
机构：
[1] Inha Univ, Dept Chem, Coll Nat Sci, Inchon 402751, South Korea
来源：
BULLETIN OF THE KOREAN CHEMICAL SOCIETY | 2012年 / 33卷 / 01期
关键词：
Isoxazol-5(4H)-one; Protein tyrosine phosphatase; Inhibitor; PTP1B; TYROSINE-PHOSPHATASE; 1B; OBESITY; STRATEGIES; RESISTANCE; ACID;
D O I：
10.5012/bkcs.2012.33.1.275
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：275 / 277
页数：3
相关论文
共 50 条
  • [21] Small Molecule Inhibitors of PTP1B and TCPTP
    Reddy, M. V. V. V. Sekhar
    Chakshusmathi, G.
    Narasu, M. Lakshmi
    INTERNATIONAL JOURNAL OF PHARMACEUTICAL AND PHYTOPHARMACOLOGICAL RESEARCH, 2012, 1 (05): : 287 - 291
  • [22] PTP1B inhibitors from Ardisia japonica
    Li, YF
    Hu, LH
    Lou, FC
    Li, J
    Shen, Q
    JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2005, 7 (01) : 13 - 18
  • [23] Identification and characterization of potent and selective inhibitors targeting protein tyrosine phosphatase 1B (PTP1B)
    Jin, Jia
    Ye, Xiaoqing
    Boateng, Derrick
    Dai, Kaili
    Ye, Fei
    Du, Pengfei
    Yu, Han
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (16) : 2358 - 2363
  • [24] Docking studies on formylchromone derivatives as protein tyrosine phosphatase 1B (PTP1B) inhibitors
    Kim, Chan Kyung
    Lee, Kyung A.
    Zhang, Hui
    Cho, Hyeongjin
    Lee, Bon-Su
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2007, 28 (07) : 1141 - 1150
  • [25] Dithiocarbamates as potential PTP1B inhibitors for diabetes management
    Deshpande, Tanvi A.
    Martinez-Malaga, Jimena
    Priefer, Ronny
    RESULTS IN CHEMISTRY, 2022, 4
  • [26] Discovery of potent PTP1B inhibitors via structure-based drug design, synthesis and in vitro bioassay of Norathyriol derivatives
    Xue, Wenjie
    Tian, Jinlong
    Wang, Xiang Simon
    Xia, Jie
    Wu, Song
    BIOORGANIC CHEMISTRY, 2019, 86 : 224 - 234
  • [27] Identification of lipid-like salicylic acid-based derivatives as potent and membrane-permeable PTP1B inhibitors
    Li, Liang
    Tavallaie, Mojdeh S.
    Xie, Fangzhou
    Xia, Yu
    Liang, Yaoyao
    Jiang, Faqin
    Fu, Lei
    BIOORGANIC CHEMISTRY, 2019, 93
  • [28] Inhibitors of protein tyrosine phosphatase 1B (PTP1B)
    Taylor, SD
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2003, 3 (07) : 759 - 782
  • [29] Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B
    Li, Xiang-Qian
    Xu, Qi
    Luo, Jiao
    Wang, Li-Jun
    Jiang, Bo
    Zhang, Ren-Shuai
    Shi, Da-Yong
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 136 : 348 - 359
  • [30] Natural PTP1B inhibitors from Broussonetia papyrifera
    Chen, RM
    Hu, LH
    An, TY
    Li, J
    Shen, Q
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2002, 12 (23) : 3387 - 3390
12345