A novel approach to homochiral beta-amino acids

被引：33
|
作者：
Seki, M
Matsumoto, K
机构：
[1] Lead Optimization Res. Laboratory, Tanabe Seiyaku Co., Ltd., Osaka 532, 16-89, Kashima-3-chome, Yodogawa-ku
来源：
TETRAHEDRON LETTERS | 1996年 / 37卷 / 18期
关键词：
D O I：
10.1016/0040-4039(96)00518-7
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient synthesis of gamma-aryl or alkyl substituted beta-amino acids starting from N-Cbz-L-homoserine lactone via the formation of alpha-amino aryl, alkenyl or alkynyl ketones with the original alpha-carbon chirality retained as such is described. Copyright (C) 1996 Elsevier Science Ltd
引用
收藏
页码：3165 / 3168
页数：4
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