1,2,3,6-Tetrahydropyrrolo[1,2-d][1,4]diazocines. Reactions of 1-methyl-2-R-tetrahydropyrrolo[1,2-a]pyrazines with alkynes

被引：1

作者：

Voskressensky, L. G. ^{[1
]}

Borisova, T. N. ^{[1
]}

Kamalitdinova, T. M. ^{[1
]}

Titov, A. A. ^{[1
]}

Listratova, A. V. ^{[1
]}

Varlamov, A. V. ^{[1
]}

机构：

[1] Peoples Friendship Univ Russia, Moscow 117198, Russia

来源：

RUSSIAN CHEMICAL BULLETIN | 2010年 / 59卷 / 03期

基金：

俄罗斯基础研究基金会;

关键词：

tetrahydropyrrolo[1,2-a]pyrazines; pyrrolo[1,2-d][1,4]diazocines; tandem transformation; ring expansion;

D O I：

10.1007/s11172-010-0119-y

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The reactions of 6-formyl- and 6-trifluoroacetyl-1-methyl-2-R-tetrahydropyrrolo[1,2-a]pyrazines with activated alkynes in methanol and acetonitrile have been studied. Terahydropyrrolo[1,2-d][1,4] diazocine derivatives were synthesized at the first time.

引用

页码：647 / 653

页数：7

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