A novel synthesis of pyrrolo[1,2-d][1,4]diazocines from tetrahydropyrrolo[1,2-a]pyrazines using activated alkynes in pyrazine ring expansion

被引：7

作者：

Voskressensky, Leonid G. ^{[1
]}

Titov, Alexander A. ^{[1
]}

Borisova, Tatiana N. ^{[1
]}

Listratova, Anna V. ^{[1
]}

Borisov, Roman S. ^{[2
]}

Kulikova, Larisa N. ^{[1
]}

Varlamov, Alexey V. ^{[1
]}

机构：

[1] Russian Peoples Friendship Univ, Dept Organ Chem, Moscow 117198, Russia

[2] Russian Acad Sci, AV Topchiev Petrochem Synth Inst, Moscow 119991, Russia

来源：

TETRAHEDRON | 2010年 / 66卷 / 27-28期

基金：

俄罗斯基础研究基金会;

关键词：

Pyrrolopyrazines; Pyrrolo[1,4]diazocines; Activate alkynes; Ring expansion; Michael addition; RECEPTOR ANTAGONISTS; DESIGN;

D O I：

10.1016/j.tet.2010.04.104

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：5140 / 5148

页数：9

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[1] First example of the synthesis of pyrrolo[1,2-d][1,4]diazocine by the reaction of tetrahydropyrrolo[1,2-a]pyrazines with activated alkynes
L. G. Voskresensky
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[J]. Chemistry of Heterocyclic Compounds, 2008, 44 : 634 - 636
[2] FIRST EXAMPLE OF THE SYNTHESIS OF PYRROLO[1,2-d][1,4]DIAZOCINE BY THE REACTION OF TETRAHYDROPYRROLO[1,2-a]PYRAZINES WITH ACTIVATED ALKYNES
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