Microwave Assisted Synthesis of 1,2,4-Triazolo[4,3-a]perimidines

被引：0
|
作者：
Davoodnia, A. [1 ]
Saeidi, A. [1 ]
Tavakoli-Hoseini, N. [1 ]
机构：
[1] Islamic Azad Univ, Mashhad Branch, Dept Chem, Mashhad, Iran
来源：
ASIAN JOURNAL OF CHEMISTRY | 2012年 / 24卷 / 05期
关键词：
1,2,4-Triazolo[4,3-a]perimidines; Cyclocondensation; Microwave irradiation; Triethylorthoesters; ANTIMICROBIAL ACTIVITY; STRUCTURE ELUCIDATION; RAPID SYNTHESIS; DERIVATIVES; IRRADIATION;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Microwave assisted synthesis of some 1,2,4-triazolo[4,3-a]perimidines through cyclocondensation reaction of 2-hydrazino-1H-perimidine I with triethylorthoesters or aryl nitriles in solvent-free conditions is described. The present methodology offers several advantages, such as a simple procedure with an easy work-up, short reaction times, high yields and the absence of any volatile and hazardous organic solvents.
引用
收藏
页码：2313 / 2316
页数：4
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