Preparation and Photosynthesis-Inhibiting Activity of 1-[(2-Chlorophenyl)carbamoyl]naphthalen-2-yl Alkylcarbamates

被引：0
|
作者：
Gonec, Tomas [1 ]
Stranik, Josef [1 ]
Pesko, Matus [2 ]
Kos, Jiri [1 ]
Oravec, Michal [3 ]
Kralova, Katarina [4 ]
Jampilek, Josef [1 ]
机构：
[1] Univ Vet & Pharmaceut Sci, Fac Pharm, Dept Chem Drugs, Palackeho 1-3, Brno 61242, Czech Republic
[2] Comenius Univ, Fac Nat Sci, Dept Environm Ecol, Bratislava 84215, Slovakia
[3] Global Change Res Ctr AS CR, Brno 60300, Czech Republic
[4] Comenius Univ, Fac Nat Sci, Inst Chem, Bratislava 84215, Slovakia
来源：
19TH INTERNATIONAL ELECTRONIC CONFERENCE ON SYNTHETIC ORGANIC CHEMISTRY | 2015年
关键词：
Alkylcarbamates; Hydroxynaphthalene-carboxamides; PET inhibition; Spinach chloroplasts; Structure-activity relationships; ELECTRON-TRANSPORT; HERBICIDAL ACTIVITY; BIOLOGICAL-ACTIVITY; SUBSTITUTED BENZANILIDES; ANTIBACTERIAL; SPECTRUM; ANTIMYCOBACTERIAL; CHLOROPLASTS; ACIDS;
D O I：
10.3390/ecsoc-19-b006
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
In this study a series of eight 1-[(2-chlorophenyl) carbamoyl] naphthalen-2-yl alkylcarbamates was prepared and characterized. The discussed compounds were prepared by microwave-assisted and conventional synthesis. The compounds were tested for their activity related to inhibition of photosynthetic electron transport (PET) in spinach (Spinacia oleracea L.) chloroplasts. The PET-inhibiting activity of the compounds was moderate; the highest activity within the series of compounds was observed for 1-[(2-chlorophenyl)-carbamoyl] naphthalen-2-yl propylcarbamate, and the compounds were found to inhibit PET in photosystem II.
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页数：10
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