GPBAR1 (TGR5) IS A MODULATOR OF LIVER IMMUNITY AND REVERSES LIVER INFLAMMATION IN A MOUSE MODELS OF ACUTE HEPATITIS

被引:0
|
作者
Biagioli, Michele
Carino, Adriana
Fiorucci, Chiara
Marchiano, Silvia
Zampella, Angela
Distrutti, Eleonora
Fiorucci, Stefano
机构
关键词
D O I
暂无
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
241
引用
收藏
页码:S1078 / S1078
页数:1
相关论文
共 50 条
  • [31] The Deficiency of G-Protein-Coupled Bile Acid Receptor Gpbar1 (TGR5) Enhances Chemically-Induced Liver Carcinogenesis (Retraction of vol 57, pg 656, 2012)
    Chen, Wei-Dong
    Yu, Donna
    Forman, Barry M.
    Huang, Wendong
    Wang, Yan-Dong
    HEPATOLOGY, 2013, 58 (03) : 1194 - 1194
  • [32] The G-Protein-Coupled Bile Acid Receptor Gpbar1 (TGR5) Inhibits Gastric Inflammation Through Antagonizing NF-κB Signaling Pathway
    Guo, Cong
    Qi, Hui
    Yu, Yingjie
    Zhang, Qiqi
    Su, Jia
    Yu, Donna
    Huang, Wendong
    Chen, Wei-Dong
    Wang, Yan-Dong
    FRONTIERS IN PHARMACOLOGY, 2015, 6
  • [33] Aberrant DNA Methylation of G-protein-coupled Bile Acid Receptor Gpbar1 (TGR5) is a Potential Biomarker for Hepatitis B Virus Associated Hepatocellular Carcinoma
    Han, Li-Yan
    Fan, Yu-Chen
    Mu, Nan-Nan
    Gao, Shuai
    Li, Feng
    Ji, Xiang-Fen
    Dou, Cheng-Yun
    Wang, Kai
    INTERNATIONAL JOURNAL OF MEDICAL SCIENCES, 2014, 11 (02): : 164 - 171
  • [34] Design of G-protein-coupled bile acid receptor 1 (GPBAR1, TGR5) soft drugs with reduced gallbladder-filling effects
    Han, Fanghui
    Ning, Mengmeng
    Cao, Hua
    Ye, Yangliang
    Feng, Ying
    Leng, Ying
    Shen, Jianhua
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 203
  • [35] BILE ACID RECEPTORS FXR AND TGR IN LIVER FIBROSIS AND INFLAMMATION: STUDY OF FXR/TGR5 DOUBLE KNOCKOUT MICE
    Ferrell, Jessica M.
    Boehme, Shannon
    Gilliland, Tricia
    Chiang, John Y. L.
    HEPATOLOGY, 2019, 70 : 1378A - 1378A
  • [36] TUDCA skews microglia towards M2 phenotype through the G-protein coupled bile acid receptor GPBAR1/TGR5
    Yanguas Casas, N.
    de la Barreda Manso, M. A.
    Nieto Sampedro, M.
    Romero Ramirez, L.
    GLIA, 2015, 63 : E357 - E357
  • [37] G-Protein-Coupled Bile Acid Receptor 1 (GPBAR1, TGR5) Agonists Reduce the Production of Proinflammatory Cytokines and Stabilize the Alternative Macrophage Phenotype
    Hoegenauer, Klemens
    Arista, Luca
    Schmiedeberg, Niko
    Werner, Gudrun
    Jaksche, Herbert
    Bouhelal, Rochdi
    Nguyen, Deborah G.
    Bhat, B. Ganesh
    Raad, Layla
    Rauld, Celine
    Carballido, Jose M.
    JOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (24) : 10343 - 10354
  • [38] Vertical sleeve gastrectomy activates GPBAR-1/TGR5 to sustain weight loss, improve fatty liver, and remit insulin resistance in mice
    Ding, Lili
    Sousa, Kyle M.
    Jin, Lihua
    Dong, Bingning
    Kim, Byung-Wook
    Ramirez, Ricardo
    Xiao, Zhenzhou
    Gu, Ying
    Yang, Qiaoling
    Wang, Jie
    Yu, Donna
    Pigazzi, Alessio
    Schones, Dustin
    Yang, Li
    Moore, David
    Wang, Zhengtao
    Huang, Wendong
    HEPATOLOGY, 2016, 64 (03) : 760 - 773
  • [39] Combinatorial therapy with BAR502 and UDCA resets FXR and GPBAR1 signaling and reverses liver histopathology in a model of NASH
    Marchiano, Silvia
    Biagioli, Michele
    Morretta, Elva
    Di Giorgio, Cristina
    Roselli, Rosalinda
    Bordoni, Martina
    Bellini, Rachele
    Urbani, Ginevra
    Massa, Carmen
    Monti, Maria Chiara
    Zampella, Angela
    Distrutti, Eleonora
    Fiorucci, Stefano
    SCIENTIFIC REPORTS, 2023, 13 (01)
  • [40] The bile acid receptor GPBAR1 (TGR5) is expressed in human gastric cancers and promotes epithelial-mesenchymal transition in gastric cancer cell lines
    Carino, Adriana
    Graziosi, Luigina
    D'Amore, Claudio
    Cipriani, Sabrina
    Marchiano, Silvia
    Marino, Elisabetta
    Zampella, Angela
    Rende, Mario
    Mosci, Paolo
    Distrutti, Eleonora
    Donini, Annibale
    Fiorucci, Stefano
    ONCOTARGET, 2016, 7 (38) : 61021 - 61035