An efficient organocatalytic method for tandem synthesis of functionalized 2-pyridones

被引：17
|
作者：
Yavari, Issa [1 ]
Bayat, Mohammad J. [1 ]
机构：
[1] Tarbiat Modares Univ, Dept Chem, Tehran, Iran
来源：
TETRAHEDRON LETTERS | 2011年 / 52卷 / 49期
关键词：
Primary amine; Acetylenic ester; 2-Pyridone; MCRs; Tandem reaction;
D O I：
10.1016/j.tetlet.2011.10.029
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Highly functionalized 2-pyridones are obtained via a tandem reaction between primary amines and acetylenic esters in the presence of N-methylimidazole as an organocatalyst. (C) 2011 Elsevier Ltd. All rights reserved.
引用
收藏
页码：6649 / 6651
页数：3
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