Direct carboxamidation of indoles by palladium-catalyzed C-H activation and isocyanide insertion

被引：102
|
作者：
Peng, Jiangling [1 ,2 ]
Liu, Lanying [1 ,2 ]
Hu, Ziwei [1 ,2 ]
Huang, Jinbo [1 ,2 ]
Zhu, Qiang [1 ,2 ]
机构：
[1] Chinese Acad Sci, State Key Lab Resp Dis, Guangzhou Inst Biomed, 190 Kaiyuan Ave, Guangzhou 510530, Guangdong, Peoples R China
[2] Chinese Acad Sci, State Key Lab Resp Dis, Guangzhou Inst Hlth, Guangzhou 510530, Guangdong, Peoples R China
来源：
CHEMICAL COMMUNICATIONS | 2012年 / 48卷 / 31期
基金：
美国国家科学基金会;
关键词：
FUNCTIONALIZATION; AMIDATION; MILD; 4-AMINOQUINAZOLINES; ALKENYLATION; HETEROARENES; ANNULATION; CYANATION; BONDS;
D O I：
10.1039/c2cc30351e
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A selective C3 carboxamidation of indoles including free (N-H) ones by palladium-catalyzed sequential C-H activation-isocyanide insertion has been developed.
引用
收藏
页码：3772 / 3774
页数：3
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