Effect of subunit composition and agonist of GABAA receptor on the noncompetitive antagonist binding

被引:0
|
作者
Chen, Ligong [1 ]
Casida, John E. [1 ]
机构
[1] Univ Calif Berkeley, Dept Environm Sci Policy & Management, Berkeley, CA 94720 USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
153
引用
收藏
页码:75 / 75
页数:1
相关论文
共 50 条
  • [31] CPCCOEt, a noncompetitive metabotropic glutamate receptor 1 antagonist, inhibits receptor signaling without affecting glutamate binding
    Litschig, S
    Gasparini, F
    Rueegg, D
    Stoehr, N
    Flor, PJ
    Vranesic, I
    Prezeau, L
    Pin, JP
    Thomsen, C
    Kuhn, R
    MOLECULAR PHARMACOLOGY, 1999, 55 (03) : 453 - 461
  • [32] Agonist trapping by GABAA receptor channels
    Bianchi, MT
    Macdonald, RL
    JOURNAL OF NEUROSCIENCE, 2001, 21 (23): : 9083 - 9091
  • [33] Allosterically linked noncompetitive antagonist binding sites in the resting nicotinic acetylcholine receptor ion channel
    Arias, HR
    McCardy, EA
    Bayer, EZ
    Gallagher, MJ
    Blanton, MP
    ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 2002, 403 (01) : 121 - 131
  • [34] Agonist-Specific Conformational Changes in the α1-γ2 Subunit Interface of the GABAA Receptor
    Eaton, Megan M.
    Lim, You Bin
    Bracamontes, John
    Steinbach, Joe Henry
    Akk, Gustav
    MOLECULAR PHARMACOLOGY, 2012, 82 (02) : 255 - 263
  • [35] Azogabazine; a photochromic antagonist of the GABAA receptor
    Huckvale, Rosemary
    Mortensen, Martin
    Pryde, David
    Smart, Trevor G.
    Baker, James R.
    ORGANIC & BIOMOLECULAR CHEMISTRY, 2016, 14 (28) : 6676 - 6678
  • [36] SOMATOSTATIN IS AN AGONIST AND NONCOMPETITIVE ANTAGONIST OF GASTRIN IN OXYNTIC CELL-FUNCTION
    SHAPIRO, B
    PIENTA, K
    HELDSINGER, A
    VINIK, AI
    ENDOCRINOLOGY, 1981, 109 (04) : 1117 - 1121
  • [37] DECIDIUM - A NOVEL FLUORESCENT-PROBE OF THE AGONIST ANTAGONIST AND NONCOMPETITIVE INHIBITOR SITES ON THE NICOTINIC ACETYLCHOLINE-RECEPTOR
    JOHNSON, DA
    BROWN, RD
    HERZ, JM
    BERMAN, HA
    ANDREASEN, GL
    TAYLOR, P
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1987, 262 (29) : 14022 - 14029
  • [38] PROTEOLYTIC MAPPING OF THE AGONIST AND ALLOSTERIC ANTAGONIST BINDING-SITES ON THE NICOTINIC ACETYLCHOLINE-RECEPTOR (ACHR) ALPHA-SUBUNIT
    PEDERSEN, SE
    DREYER, EB
    COHEN, JB
    BIOPHYSICAL JOURNAL, 1986, 49 (02) : A361 - A361
  • [39] Involvement of GABAA receptor-associated chloride channels in the peripheral antinociceptive effect induced by GABAA receptor agonist muscimol
    Reis, Glaucia
    Pacheco, Daniela
    Francischi, Janetti
    Castro, Maria
    Perez, Andrea
    Duarte, Igor
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2007, 564 (1-3) : 112 - 115
  • [40] THERMODYNAMIC ANALYSIS OF AGONIST AND ANTAGONIST BINDING TO THE CHICKEN BRAIN MELATONIN RECEPTOR
    CHONG, NWS
    SUGDEN, D
    BRITISH JOURNAL OF PHARMACOLOGY, 1994, 111 (01) : 295 - 301