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- [1] Development of Highly Potent and Selective Covalent FGFR4 Inhibitors Based on SNAr Electrophiles[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (08) : 6549 - 6569Schwarz, Moritz论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyKurkunov, Maksym论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & Fu, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyWittlinger, Florian论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyRudalska, Ramona论文数: 0 引用数: 0 h-index: 0机构: Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & Fu, D-72076 Tubingen, Germany Univ Hosp Tubingen, Dept Med Oncol & Pneumol, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyWang, Guiqun论文数: 0 引用数: 0 h-index: 0机构: German Canc Res Ctr, German Canc Res Consortium DKTK, D-69120 Heidelberg, Germany Goethe Univ Frankfurt, Buchmann Inst Mol Life Sci, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt, Inst Pharmaceut Chem, D-60438 Frankfurt, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany论文数: 引用数: h-index:机构:Rasch, Alexander论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyWagner, Benedikt论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & Fu, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyLaufer, Stefan A.论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & Fu, D-72076 Tubingen, Germany Tubingen Ctr Acad Drug Discovery & Dev TuCAD2, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyKnapp, Stefan论文数: 0 引用数: 0 h-index: 0机构: German Canc Res Ctr, German Canc Res Consortium DKTK, D-69120 Heidelberg, Germany Goethe Univ Frankfurt, Buchmann Inst Mol Life Sci, Struct Genom Consortium SGC, D-60438 Frankfurt, Germany Goethe Univ Frankfurt, Inst Pharmaceut Chem, D-60438 Frankfurt, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyDauch, Daniel论文数: 0 引用数: 0 h-index: 0机构: Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & Fu, D-72076 Tubingen, Germany Univ Hosp Tubingen, Dept Med Oncol & Pneumol, D-72076 Tubingen, Germany Tubingen Ctr Acad Drug Discovery & Dev TuCAD2, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyGehringer, Matthias论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & Fu, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Inst Pharmaceut Sci, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany
- [2] Discovery of Selective, Covalent FGFR4 Inhibitors with Antitumor Activity in Models of Hepatocellular Carcinoma[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2020, 11 (10): : 1899 - 1904Liu, Haibo论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USANiu, Deqiang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USASjin, Robert Tjin Tham论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USADubrovskiy, Alex论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAZhu, Zhendong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAMcDonald, Joseph J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAFahnoe, Kelly论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAWang, Zhigang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAMunson, Mark论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAScholte, Andrew论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USABarrague, Matthieu论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAFitzgerald, Maria论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USALiu, Jinyu论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAKothe, Michael论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USASun, Fangxian论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAMurtie, Joshua论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAGe, Jie论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USARocnik, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAHarvey, Darren论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAOspina, Beatriz论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAPerron, Keli论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAZheng, Gang论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAShehu, Elvis论文数: 0 引用数: 0 h-index: 0机构: Dept Integrated Drug Discovery, Waltham, MA 02451 USA Dept DMPK, Waltham, MA 02451 USA Dept Pharmacol, Waltham, MA 02451 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USAD'Agostino, Laura Akullian论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biol, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Biochem, Cambridge, MA 02140 USA Bristol Myers Squibb, Dept Chem, Cambridge, MA 02140 USA
- [3] Design, synthesis, and biological evaluation of selective covalent inhibitors of FGFR4[J]. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 268Chen, Xiaojuan论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaLi, Huiliang论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Chem & Chem Engn, Key Lab Chem Biol & Tradit Chinese Med, Minist Educ China,Key Lab Assembly & Applicat Orga, Changsha, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaLin, Qianmeng论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaDai, Shuyan论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Sch Pharmaceut Sci, Dept Pharmacol, Changsha 410078, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaQu, Lingzhi论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaGuo, Ming论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaZhang, Lin论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaLiao, Jiaxuan论文数: 0 引用数: 0 h-index: 0机构: HD Shanghai Sch, Shanghai 201613, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaWei, Hudie论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaXu, Guangyu论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Chem & Chem Engn, Key Lab Chem Biol & Tradit Chinese Med, Minist Educ China,Key Lab Assembly & Applicat Orga, Changsha, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaJiang, Longying论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Pathol, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R ChinaChen, Yongheng论文数: 0 引用数: 0 h-index: 0机构: Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Natl Clin Res Ctr Geriatr Disorders, Changsha 410008, Hunan, Peoples R China Cent South Univ, Xiangya Hosp, Dept Oncol, NHC Key Lab Canc Prote,State Local Joint Engn Lab, Changsha 410008, Hunan, Peoples R China
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