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- [1] Discovery of highly potent, selective, covalent inhibitors of JAK3[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 27 (20) : 4622 - 4625Kempson, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAOvalle, Damaso论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAGuo, Junqing论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAWrobleski, Stephen T.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USALin, Shuqun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USASpergel, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USADuan, James J. -W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAJiang, Bin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USALu, Zhonghui论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USADas, Jagabandhu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAYang, Bingwei V.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAHynes, John, Jr.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USATokarski, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USASack, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAKhan, Javed论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USASchieven, Gary论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USABlatt, Yuval论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAChaudhry, Charu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USASalter-Cid, Luisa M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAFura, Aberra论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USABarrish, Joel C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USACarter, Percy H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAPitts, William J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA
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- [4] Discovery of a Highly Potent, Selective Reversible Covalent Inhibitor of JAK3 Kinase[J]. ARTHRITIS AND RHEUMATISM, 2012, 64 (10): : S982 - S982Hill, Ronald J.论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USABisconte, Angelina论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USABradshaw, J. Michael论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USABrameld, Ken论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USAKim, Eun Ok论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USALi, Xiaoyan论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USAOwens, Tim论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USAVerner, Erik论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USAGoldstein, David M.论文数: 0 引用数: 0 h-index: 0机构: Principia Biopharma, San Francisco, CA USA Principia Biopharma, San Francisco, CA USA
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h-index: 0机构: Merck KGaA, Frankfurter Str 250, DE-64293 Darmstadt, Hessen, Germany EMD Serono Res & Dev Inst, 45A Middlesex Turnpike, Billerica, MA 01821 USAGardberg, Anna论文数: 0 引用数: 0 h-index: 0机构: Constellat Pharmaceut, 215 First St 200, Cambridge, MA 02142 USA EMD Serono Res & Dev Inst, 45A Middlesex Turnpike, Billerica, MA 01821 USAGlaser, Nina论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Frankfurter Str 250, DE-64293 Darmstadt, Hessen, Germany EMD Serono Res & Dev Inst, 45A Middlesex Turnpike, Billerica, MA 01821 USAGoettsche, Anja论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, Frankfurter Str 250, DE-64293 Darmstadt, Hessen, Germany EMD Serono Res & Dev Inst, 45A Middlesex Turnpike, Billerica, MA 01821 USAGoutopoulos, Andreas论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst, 45A Middlesex Turnpike, Billerica, MA 01821 USA EMD Serono Res & Dev Inst, 45A Middlesex Turnpike, Billerica, MA 01821 USAGrenningloh, Roland论文数: 0 引用数: 0 h-index: 0机构: EMD Serono Res & Dev Inst, 45A Middlesex 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